Compile Data Set for Download or QSAR
maximum 50k data
Found 1952 with Last Name = 'ullrich' and Initial = 't'
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.0300nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  0.680nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50221416(22-methyl-(2S,13R)-14-oxa-11,22-diazaheptacyclo[13...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  0.940nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  1.20nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473905(CHEMBL130814)
Affinity DataKi:  1.89nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473905(CHEMBL130814)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098677(17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  3.20nMAssay Description:Antagonist activity of compound on SNC 80 stimulated [35S]GTP-gamma-S binding to delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098683(17-(2-methylpropyl)-6,7-dehydro-4,5alpha-epoxy-3,1...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  4.30nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  4.70nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105774(22-(2-methylallyl)-(2S,13R)-14-oxa-11,22-diazahept...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473904(CHEMBL2112670)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098676(17-(3-methylbutyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105776(22-(2-methylallyl)-(2S,13R)-11,14-dioxa-22-azahept...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098681(17-butyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098675(17-pentyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105772(6-(4-chlorophenyl)-19-(2-methylallyl)-(2S,10R)-11-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098679(17-(3-methyl-2-butenyl)-6,7-dehydro-4,5alpha-epoxy...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098672(17-hexyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  30nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098678(17-(1-methylethyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105782(18-(2-methylallyl)-(2S,9R)-10-oxa-6,7,18-triazahex...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105782(18-(2-methylallyl)-(2S,9R)-10-oxa-6,7,18-triazahex...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105777(17-(2-methylallyl)-substituted noroxymorphone deri...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105773(17-(2-methylallyl)-substituted noroxymorphone deri...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473907(CHEMBL2112671)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50221416(22-methyl-(2S,13R)-14-oxa-11,22-diazaheptacyclo[13...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]DAMGO at mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098682(17-heptyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]DADLE at delta-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098674((E)-17-(2-butenyl)-6,7-dehydro-4,5alpha-epoxy-3,14...)
Affinity DataKi:  118nMAssay Description:Antagonist activity of compound on U50,488H stimulated [35S]GTP-gamma-S binding to opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105782(18-(2-methylallyl)-(2S,9R)-10-oxa-6,7,18-triazahex...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]DAMGO from Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473906(CHEMBL2111861)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098673(17-(2-methyl-2-propenyl)-6,7-dehydro-4,5alpha-epox...)
Affinity DataKi:  200nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105780(10,17-dihydroxy-4-(2-methylallyl)-15-[1-phenyl-(E)...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105771(6-(4-chlorophenyl)-13-methoxy-19-(2-methylallyl)-(...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098680(17-ethyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydroxy...)
Affinity DataKi:  290nMAssay Description:Antagonist activity of compound on DAMGO stimulated [35S]GTP-gamma-S binding to mu-opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105772(6-(4-chlorophenyl)-19-(2-methylallyl)-(2S,10R)-11-...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]U-69593 from Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50098677(17-propyl-6,7-dehydro-4,5alpha-epoxy-3,14-dihydrox...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]U-69593 at opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50105775(16-methoxy-22-(2-methylallyl)-(2S,13R)-14-oxa-11,2...)
Affinity DataKi:  500nMAssay Description:Displacement of [3H]DADLE from Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Vienna University Of Technology

Curated by ChEMBL
LigandPNGBDBM50473910(CHEMBL2111860)
Affinity DataKi:  533nMAssay Description:Displacement of [3H]cytisine from Nicotinic acetylcholine receptor alpha4-beta2 in rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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