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Found 87 with Last Name = 'ustyugov' and Initial = 'aa'
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262661(CHEMBL4075825)
Affinity DataKi:  160nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262660(CHEMBL4065259)
Affinity DataKi:  350nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262687(CHEMBL4077169)
Affinity DataKi:  410nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262637(CHEMBL4088659)
Affinity DataKi:  490nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262651(CHEMBL4080726)
Affinity DataKi:  940nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262656(CHEMBL4067342)
Affinity DataKi:  1.46E+3nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262666(CHEMBL4104952)
Affinity DataKi:  2.66E+3nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262661(CHEMBL4075825)
Affinity DataKi:  3.34E+3nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262660(CHEMBL4065259)
Affinity DataKi:  3.75E+3nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262687(CHEMBL4077169)
Affinity DataKi:  4.01E+3nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262637(CHEMBL4088659)
Affinity DataKi:  6.43E+3nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262651(CHEMBL4080726)
Affinity DataKi:  1.32E+4nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262666(CHEMBL4104952)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  29nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262687(CHEMBL4077169)
Affinity DataIC50:  460nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262661(CHEMBL4075825)
Affinity DataIC50:  810nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262660(CHEMBL4065259)
Affinity DataIC50:  840nMAssay Description:Negative allosteric modulation of rat mGlu5 receptor expressed in HEK293 cells assessed as inhibition of glutamate induced-calcium mobilization prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262637(CHEMBL4088659)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262662(CHEMBL4075624)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50130915(CHEBI:3122 | CHEMBL1231178)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262656(CHEMBL4067342)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262651(CHEMBL4080726)
Affinity DataIC50:  3.35E+3nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262640(CHEMBL4063635)
Affinity DataIC50:  4.83E+3nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262666(CHEMBL4104952)
Affinity DataIC50:  7.62E+3nMAssay Description:Competitive inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by L...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262660(CHEMBL4065259)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262687(CHEMBL4077169)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262637(CHEMBL4088659)
Affinity DataIC50:  1.24E+4nMAssay Description:Competitive inhibition of human serum AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by Lineweaver-Burk double re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262638(CHEMBL4074993)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262655(CHEMBL4096311)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262636(CHEMBL4083288)
Affinity DataIC50:  1.57E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262662(CHEMBL4075624)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262661(CHEMBL4075825)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262652(CHEMBL4097249)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262648(CHEMBL4102576)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262647(CHEMBL4077493)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262646(CHEMBL4094837)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262645(CHEMBL4087149)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262644(CHEMBL4103528)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262642(CHEMBL4080800)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262638(CHEMBL4074993)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262636(CHEMBL4083288)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human erythrocyte AChE using acetylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262656(CHEMBL4067342)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262660(CHEMBL4065259)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262658(CHEMBL4091935)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262652(CHEMBL4097249)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262691(CHEMBL4084629)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of pig liver carboxylesterase using 4-nitrophenol acetate as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262688(CHEMBL4071110)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262686(CHEMBL4078265)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Institute Of Physiologically Active Compounds Russian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50262691(CHEMBL4084629)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by substrate addition by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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