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Found 79 with Last Name = 'varnavas' and Initial = 'a'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-BH-JMV-179 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-SR-27897 from wild type human CCK1 receptor expressed in COS7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  59.8nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  169nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  973nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK1 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataKi:  1.53E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [125I]BH-(Thr,-Nle)-CCK-9 from human CCK2 receptor expressed in COS-7 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360276(CHEMBL1933104)
Affinity DataIC50:  9.5nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360273(CHEMBL1933100)
Affinity DataIC50:  15.7nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278373(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  27nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278305(2(R)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoylamin...)
Affinity DataIC50:  46nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278071(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  52nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298593((R)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278817(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  83nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278072(2-(R,S)-{2-[(1-Methyl-1H-indole-2-carbonyl)-amino]...)
Affinity DataIC50:  92nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298576((R)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-phe...)
Affinity DataIC50:  106nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360274(CHEMBL1933101)
Affinity DataIC50:  107nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298589((R)-2-(2-(5-fluoro-1H-indole-2-carboxamido)benzami...)
Affinity DataIC50:  151nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298592((+/-)-2-(2-(7-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  159nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185261(4-(3,4-dichlorobenzamido)-5-((3-methoxypropyl)(pen...)
Affinity DataIC50:  195nMAssay Description:Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  197nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278816(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  288nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298591((+/-)-2-(2-(6-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  294nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360275(CHEMBL1933103)
Affinity DataIC50:  313nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298588((+/-)-2-(2-(5-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  314nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360272(CHEMBL1933099)
Affinity DataIC50:  317nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298579((+/-)-2-(2-(1-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  350nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360277(CHEMBL1933108)
Affinity DataIC50:  419nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278135(2-(R,S)-{2-[(1H-Indole-2-carbonyl)-amino]-benzoyla...)
Affinity DataIC50:  445nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298583((+/-)-3-phenyl-2-(2-(7-(trifluoromethyl)-1H-indole...)
Affinity DataIC50:  538nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298582((+/-)-2-(2-(7-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  671nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50360278(CHEMBL1933109)
Affinity DataIC50:  717nMAssay Description:Displacement of [125I]-BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acini after 120 hrs by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298595((+/-)-2-(2-(benzofuran-2-carboxamido)benzamido)-3-...)
Affinity DataIC50:  891nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298587((+/-)-2-(2-(4-fluoro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  937nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298586((+/-)-2-(2-(1-methyl-5-nitro-1H-indole-2-carboxami...)
Affinity DataIC50:  1.11E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298596((+/-)-2-(2-(benzo[b]thiophene-2-carboxamido)benzam...)
Affinity DataIC50:  1.12E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278199((2R,S)-3-(4-Benzyloxy-phenyl)-2-{2-[(1H-indole-2-c...)
Affinity DataIC50:  1.16E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298572((+/-)-3-phenyl-2-(2-(4,5,6,7-tetrahydro-1H-indole-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298584((+/-)-2-(2-(5-chloro-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  1.84E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298577((+/-)-2-(2-(1H-indole-3-carboxamido)benzamido)-3-p...)
Affinity DataIC50:  1.87E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50298581((+/-)-2-(2-(3-methyl-1H-indole-2-carboxamido)benza...)
Affinity DataIC50:  2.06E+3nMAssay Description:Displacement of [125I]-CCK8 from CCK1 receptor in rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50278198((2R,S)-3-(4-Hydroxy-phenyl)-2-{2-[(1H-indole-2-car...)
Affinity DataIC50:  2.07E+3nMAssay Description:Displacement of [125I]BH-CCK8 from CCK1 receptor in Sprague-Dawley rat pancreatic acinar cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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