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Found 64 with Last Name = 'vassallo' and Initial = 'a'
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492754(CHEMBL2413568)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human Hsp90 ATPase activity assessed as inhibition of ATP hydrolysis after 60 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492753(CHEMBL2413570)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human Hsp90 ATPase activity assessed as inhibition of ATP hydrolysis after 60 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492759(CHEMBL2413569)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human Hsp90 ATPase activity assessed as inhibition of ATP hydrolysis after 60 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428820(CHEMBL2335722)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant PlGF-1/VEGFR-1 (unknown origin) interaction after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492762(CHEMBL2413565)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human Hsp90 ATPase activity assessed as inhibition of ATP hydrolysis after 60 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428820(CHEMBL2335722)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of recombinant VEGF-A/VEGFR-1 (unknown origin) interaction after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492755(CHEMBL2413587)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human Hsp90 ATPase activity assessed as inhibition of ATP hydrolysis after 60 mins by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428819(GERANIN B)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of recombinant VEGF-A/VEGFR-1 (unknown origin) interaction after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293293(6alpha,8alpha-dihydroxy-23-oxo-labd-13(14),17-dien...)
Affinity DataKd:  810nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293294(6alpha,8alpha,15(S)-trihydroxy-23-oxo-labd-13(14),...)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293295(6alpha,8alpha,15(S)-trihydroxy-23-carbossimethylla...)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293296(6alpha,8alpha-dihydroxy-23-carbossi-labd-13(14),17...)
Affinity DataKd:  7nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293297(6alpha,8alpha,15(S)-trihydroxy-23-carbossi-labd-13...)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293298(6alpha,8alpha,23-trihydroxy-labd-13(14),17-dien-16...)
Affinity DataKd:  72nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293299(6alpha,8alpha,15(S),23-tetrahydroxy-labd-13(14),17...)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293300(8alpha-hydroxy,23alpha-O-ethyl-23,6alpha-epoxy-lab...)
Affinity DataKd:  73nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293301(8alpha,15(S)-dihydroxy,23alpha-O-ethyl-23,6alpha-e...)
Affinity DataKd:  960nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin--tyrosine ligase(Homo sapiens (Human))
Universita Di Salerno

Curated by ChEMBL
LigandPNGBDBM50293302(8alpha,15(S),23alpha-trihydroxy-23,6alpha-epoxy-la...)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to TTL by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429448(CHEMBL2332347 | Catalpin)
Affinity DataKd:  5.93E+3nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429449(CHEMBL2332356 | Rehmaglutin A)
Affinity DataKd:  2.39E+3nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429450(VERMINOSIDE)
Affinity DataKd:  348nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM15359((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14-...)
Affinity DataKd:  326nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429451(CHEMBL2332366)
Affinity DataKd:  139nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429452(CHEMBL2332361)
Affinity DataKd:  73nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429453(Argenteoside B | CHEMBL2332353)
Affinity DataKd:  50nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429454(CHEMBL2332346)
Affinity DataKd:  31nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429455(CHEMBL2332355 | Specioside)
Affinity DataKd:  26nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429456(3,4-Dihydrocatalposide | CHEMBL2332365)
Affinity DataKd:  16nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429457(Argenteoside A | CHEMBL2332352)
Affinity DataKd:  14nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50429458(CHEMBL2332354 | Catalposide)
Affinity DataKd:  12nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50347503(RADICICOL)
Affinity DataKd:  4.20nMAssay Description:Binding affinity to recombinant Hsp90 alpha (unknown origin) by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50129952(2-(3-(5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-c...)
Affinity DataKd:  17nMAssay Description:Binding affinity to recombinant VEGFA (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428821(PROANTHOCYANIDIN A1)
Affinity DataKd:  476nMAssay Description:Binding affinity to recombinant VEGFA (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428819(GERANIN B)
Affinity DataKd:  48nMAssay Description:Binding affinity to recombinant VEGFA (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428820(CHEMBL2335722)
Affinity DataKd:  16nMAssay Description:Binding affinity to recombinant VEGFA (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlacenta growth factor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50129952(2-(3-(5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4H-c...)
Affinity DataKd:  8.20nMAssay Description:Binding affinity to recombinant PIGF1 (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlacenta growth factor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428821(PROANTHOCYANIDIN A1)
Affinity DataKd:  394nMAssay Description:Binding affinity to recombinant PIGF1 (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlacenta growth factor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428819(GERANIN B)
Affinity DataKd:  23nMAssay Description:Binding affinity to recombinant PIGF1 (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlacenta growth factor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50428820(CHEMBL2335722)
Affinity DataKd:  11nMAssay Description:Binding affinity to recombinant PIGF1 (unknown origin) measured for 60 seconds by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492756(CHEMBL2413566)
Affinity DataKd:  72nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492757(CHEMBL2413581)
Affinity DataKd:  89nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492758(CHEMBL2413580)
Affinity DataKd:  107nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492759(CHEMBL2413569)
Affinity DataKd:  2.80nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492755(CHEMBL2413587)
Affinity DataKd:  84nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492760(CHEMBL2413586)
Affinity DataKd:  191nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492761(CHEMBL2413582)
Affinity DataKd:  201nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492753(CHEMBL2413570)
Affinity DataKd:  3.5nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492762(CHEMBL2413565)
Affinity DataKd:  55nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM227589(Radicicol)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50492763(CHEMBL2413573)
Affinity DataKd:  237nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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