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Found 36 with Last Name = 'vesey' and Initial = 'dr'
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  2.85nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C beta type(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of Protein kinase C gamma (PKC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C beta type(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of Protein kinase C betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C beta type(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  28nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112960((1S,3R)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  30.5nMAssay Description:Inhibition of Protein kinase C betaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C gamma type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  36.5nMAssay Description:Inhibition of Protein kinase C gamma (PKC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C epsilon type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10a-hexahydro-1...)
Affinity DataIC50:  48nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112980((1R,3R)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50:  105nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112966(CHEMBL2372049 | EPQpYEEIPIYL)
Affinity DataIC50:  360nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112959(CHEMBL29298 | Phosphoric acid mono-(4-{(S)-2-acety...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112973(CHEMBL418579 | Phosphoric acid mono-[4-((S)-2-acet...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112974(CHEMBL29820 | Phosphoric acid mono-(4-{(S)-2-acety...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112975(CHEMBL282111 | Phosphoric acid mono-(4-{(S)-2-acet...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112971(CHEMBL418027 | Phosphoric acid mono-(4-{(S)-2-acet...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112968(CHEMBL413761 | Phosphoric acid mono-{4-[(S)-2-acet...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112958(CHEMBL281685 | Phosphoric acid mono-(4-{(S)-2-acet...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112964(CHEMBL29564 | Phosphoric acid mono-(4-{(S)-2-acety...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112972((S)-4-{(S)-2-[(S)-2-Acetylamino-3-(4-phosphonooxy-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112969(CHEMBL286989 | Phosphoric acid mono-{4-[(S)-2-acet...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112970(CHEMBL30157 | Phosphoric acid mono-(4-{(S)-2-acety...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112981(CHEMBL28638 | Phosphoric acid mono-{4-[(S)-2-acety...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112961(CHEMBL29139 | Phosphoric acid mono-[4-((S)-2-acety...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50366781(CHEMBL1790100)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112979((1S,3S)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112962((1R,3S)-3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phos...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112976(CHEMBL416938 | Phosphoric acid mono-{4-[(S)-2-acet...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112977(3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phosphonooxy...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112977(3-({(1S,9S)-9-[(S)-2-Acetylamino-3-(4-phosphonooxy...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112965(CHEMBL441774 | Phosphoric acid mono-{4-[(S)-2-acet...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112963(CHEMBL29723 | Phosphoric acid mono-(4-{(S)-2-acety...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112957((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Roche Products

Curated by ChEMBL
LigandPNGBDBM50112967((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  3.50E+5nMAssay Description:Inhibitory activity towards p56 Lck tyrosine kinase SH2 domain using scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed