TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (3)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 4.66nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (3)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (3)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (3)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (2)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 16.3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (2)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 21.7nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (2)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (2)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 36.6nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Cholinergic interactions was measured as displaced [3H]cystine from Nicotinic acetylcholine receptor alpha4-beta2 in rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (2)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in rat brain homogenate using 3- arylpropenyl-8-propionyl-DBO derivative (3)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Inhibition of [3H]-DAMGO binding to rat brain homogenat Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 750nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determined in guinea pig homogenate using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 2.27E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in rat brain homogenate using [3H]-deltorphin II as radioligandMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute Of Oncology
Curated by ChEMBL
European Institute Of Oncology
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibitory activity against beta-glucosidase of sweet almondMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determined in guinea pig homogenate using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:Cholinergic interactions was measured as displaced [3H]cystine from Nicotinic acetylcholine receptor alpha4-beta2 in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: 7.50E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in rat brain homogenate using [3H]-deltorphin II as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in rat brain homogenate using [3H]-deltorphin II as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Istituto Di Chimica Farmaceutica E Tossicologica
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor kappa 1 was determined in guinea pig homogenate using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute Of Oncology
Curated by ChEMBL
European Institute Of Oncology
Curated by ChEMBL
Affinity DataKi: 4.30E+4nMAssay Description:Non-competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated fo...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute Of Oncology
Curated by ChEMBL
European Institute Of Oncology
Curated by ChEMBL
Affinity DataKi: 4.84E+4nMAssay Description:Competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated for 15...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.270nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute Of Oncology
Curated by ChEMBL
European Institute Of Oncology
Curated by ChEMBL
Affinity DataIC50: 0.380nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Sapienza University Of Rome
Curated by ChEMBL
Sapienza University Of Rome
Curated by ChEMBL
Affinity DataIC50: 0.380nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute Of Oncology
Curated by ChEMBL
European Institute Of Oncology
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using biotinylated H3K4me1 peptide as substrate preincubated for 2...More data for this Ligand-Target Pair