Affinity DataIC50: 10nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 31.6nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 50.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of rat P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of rat P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
TargetBromodomain adjacent to zinc finger domain protein 2A(Homo sapiens (Human))
Gsk
Curated by ChEMBL
Gsk
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of BAZ2A (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from recombinant human N-terminal His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant incubated...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human P2X7 receptor assessed as inhibition of ethidium bromide accumulationMore data for this Ligand-Target Pair