TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.178nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in HEK293T cell homogenates incubated for 1 hr by radioligand binding assay based liquid scin...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.178nMAssay Description:Displacement of [3H]mepyramine from human histamine H1 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.251nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.398nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.417nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 0.501nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.631nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 0.631nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]NAMH from mouse H3R expressed in HEK293T cells incubated for 2 hrs by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.02nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.05nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.15nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]granisetron from human 5-HT3AR expressed in HEK293 cells after 24 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 1.62nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 2.09nMAssay Description:Displacement of [3H]mepyramine from human histamine H1 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
Affinity DataKi: 2.82nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]histamine displacement from human recombinant histamine H4 receptor expressed in SK-NM-C cells after 45 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]histamine displacement from human recombinant histamine H4 receptor expressed in SK-NM-C cells after 45 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]histamine displacement from human recombinant histamine H4 receptor expressed in SK-NM-C cells after 45 minsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]NAMH from human H3R expressed in HEK293T cells incubated for 2 hrs by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in HEK293T cells by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.68nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]histamine from human H3 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]mepyramine from N-terminal HA-tagged H1R (unknown origin) expressed in HEK293T cells measured after 4 hrs by microbeta scintillat...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]mepyramine from human wild type N-terminal hemagglutinin-tagged histamine H1 receptor expressed in HEK293T cells after 4 hrs by m...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
University Of Nottingham Biodiscovery Institute
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]mepyramine from human histamine H1 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]histamine displacement from human histamine H4 receptor expressed in SK-NM-C cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]histamine displacement from human recombinant histamine H4 receptor expressed in SK-NM-C cells after 45 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]NAMH from human H3R expressed in HEK293T cells incubated for 2 hrs by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Displacement of [3H]histamine from human H4R receptor expressed in HEK293 cells at 10 uM after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair