Affinity DataKi: 17nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1A receptor expressed in human CHO cell membranes incubated for 60 mins by scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Displacement of [3H]ZM241385 from adenosine A2A receptor in human HeLa cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity to Mcl-1More data for this Ligand-Target Pair
Affinity DataKi: 1.38E+5nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 1.39E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 1.95E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 1.16E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 1.04E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataEC50: 4.56E+3nMAssay Description:Effective concentration against DNA topoisomerase IMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+5nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 4.30E+6nMAssay Description:Inhibition of GST-tagged Bcl-xL (unknown origin) measured after 1 hr incubation by fluorescence polarization assayMore data for this Ligand-Target Pair