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PDB Reactome pathway
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583877(CHEMBL5070261)

Ki: 0.300nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583878(CHEMBL5074709)

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583879(CHEMBL5070075)

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
National Institutes Of Health

Curated by ChEMBL

BDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)

Ki: 0.340nMAssay Description:Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]-GTP-gammaS, binding (Experi...More data for this Ligand-Target Pair

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PDB Reactome pathway
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583881(CHEMBL5081323)

Ki: 0.400nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL

BDBM50076428(4-Fluoro-cyclohexanecarboxylic acid {2-[4-(2-metho...)

Ki: 0.515nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair

Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM50374600(CHEMBL272899)

Ki: 0.560nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL

BDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)

Ki: 0.590nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair

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PDB Reactome pathway
UniProtKB/SwissProt
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50546439(Balovaptan | RG-7314 | RO-5285119 | RO5285119 | Rg...)

Ki: 0.700nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

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PDB Reactome pathway
UniProtKB/SwissProt
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5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL

BDBM50076429(4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl...)

Ki: 0.791nMAssay Description:In vitro inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptor (Experiment 2)More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50546436(CHEMBL4799793)

Ki: 0.800nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM50398057(CHEMBL2181924)

Ki: 0.960nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM50398057(CHEMBL2181924)

Ki: 0.960nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair

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PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
National Institutes Of Health

Curated by ChEMBL

BDBM50076428(4-Fluoro-cyclohexanecarboxylic acid {2-[4-(2-metho...)

Ki: 1nMAssay Description:Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]-GTP-gammaS, bindingMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Vasopressin V2 receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)

Ki: 1nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V2 receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindin...More data for this Ligand-Target Pair

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PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
National Institutes Of Health

Curated by ChEMBL

BDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)

Ki: 1.10nMAssay Description:Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]GTP-gamma-S, binding (Experi...More data for this Ligand-Target Pair

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PDB Reactome pathway
UniProtKB/SwissProt
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5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL

BDBM50076429(4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl...)

Ki: 1.10nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptor (Expe...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Stanford University

Curated by ChEMBL

BDBM50338990(1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piper...)

Ki: 1.70nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair

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Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM50374600(CHEMBL272899)

Ki: 1.70nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
National Institutes Of Health

Curated by ChEMBL

BDBM50076429(4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl...)

Ki: 2.90nMAssay Description:Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]-GTP-gammaS, binding (Experi...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295040(5-(4-Cyclopropylphenyl)-1-(2-chloro-4-bromophenyl)...)

Ki: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295029(5-(4-Cyclopropylphenyl)-1-(2,4-dichlorophenyl)-4-m...)

Ki: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295024(5-(4-Cyclopropylphenyl)-1-(2,4-dichlorophenyl)-4-m...)

Ki: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)

Ki: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair

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3D Structure (crystal)

Sigma non-opioid intracellular receptor 1(RAT)
Stanford University

Curated by ChEMBL

BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)

Ki: 3.40nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair

PDB Reactome pathway
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Details Article PubMed PDB

3D Structure (crystal)

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50354894(CHEMBL1837037)

Ki: 3.5nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

CHEMBL PC cid PC sid Patents Similars

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

5-hydroxytryptamine receptor 1D(Mus musculus (Mouse))
National Institutes Of Health

Curated by ChEMBL

BDBM50076429(4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl...)

Ki: 4nMAssay Description:Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]GTP-gamma-S, bindingMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295039(5-(4-Cyclopropylphenyl)-1-(2,4-dichlorophenyl)-4-e...)

Ki: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institutes Of Health

Curated by ChEMBL

BDBM50076429(4-Fluoro-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl...)

Ki: 4nMAssay Description:Compound was tested in vitro for the inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptor (Expe...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295041(5-(4-Cyclopropylphenyl)-1-(2,4-dichlorophenyl)-4-e...)

Ki: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295032(5-(4-Cyclopropylphenyl)-1-(2-chlorophenyl)-4-methy...)

Ki: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50077217(CHEMBL3416885)

Ki: 5.5nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

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PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)

Ki: 6nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

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PDB Reactome pathway
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Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583883(CHEMBL5078950)

Ki: 6.30nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583883(CHEMBL5078950)

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)

Ki: 6.5nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair

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PDB Reactome pathway KEGG
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Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295025(5-(4-Cyclobutylphenyl)-1-(2,4-dichlorophenyl)-4-me...)

Ki: 7nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295033(5-(4-Cyclopropylphenyl)-1-(2-chloro-4-fluorophenyl...)

Ki: 8nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583880(CHEMBL5088219)

Ki: 8.80nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295034(5-(4-Cyclopropylphenyl)-1-(2-fluorophenyl)-4-methy...)

Ki: 11nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

Vasopressin V1a receptor(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL

BDBM50583887(CHEMBL5074961)

Ki: 12nMAssay Description:Displacement of [3H]-arginine-vasopressin from human V1A receptor expressed in human 1321N1 cell membranes incubated for 60 mins by radioligand bindi...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))
Anadolu University

Curated by ChEMBL

BDBM50552011(CHEMBL4792992)

Ki: 13nMAssay Description:Inhibition of human erythrocyte CA2 using 4-nitrophenyl acetate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair

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PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295027(5-(4-Cyclohexylphenyl)-1-(2,4-dichlorophenyl)-4-me...)

Ki: 13nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295037(5-(4-Cyclopropylphenyl)-1-(2-fluoro-4-chlorophenyl...)

Ki: 14nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295026(5-(4-Cyclopentylphenyl)-1-(2,4-dichlorophenyl)-4-m...)

Ki: 15nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

Cannabinoid receptor 1(Rattus norvegicus (rat))
Gedeon Richter

Curated by ChEMBL

BDBM50295028(5-(4-Cyclopropylphenyl)-1-(2,4-dichlorophenyl)-N-p...)

Ki: 16nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))
Anadolu University

Curated by ChEMBL

BDBM50552018(CHEMBL4764100)

Ki: 21nMAssay Description:Inhibition of human erythrocyte CA2 using 4-nitrophenyl acetate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))
Anadolu University

Curated by ChEMBL

BDBM50552012(CHEMBL4786423)

Ki: 26nMAssay Description:Inhibition of human erythrocyte CA2 using 4-nitrophenyl acetate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Carbonic anhydrase 2(Homo sapiens (Human))
Anadolu University

Curated by ChEMBL

BDBM50552009(CHEMBL4747356)

Ki: 28nMAssay Description:Inhibition of human erythrocyte CA2 using 4-nitrophenyl acetate as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair