Affinity DataKi: 2.40E+3nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 3.82E+3nM IC50: 2.80E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 5.67E+3nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 7.89E+3nM IC50: 8.13E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 8.22E+3nM IC50: 8.80E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 9.23E+3nM IC50: 1.12E+4nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 9.60E+3nM IC50: 8.56E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 9.70E+3nM IC50: 7.90E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 1.19E+4nM IC50: 9.33E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 1.24E+4nM IC50: 1.45E+4nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 1.36E+4nM IC50: 7.60E+3nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 1.48E+4nM IC50: 1.78E+4nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nM IC50: 2.10E+4nMpH: 6.8Assay Description:Reaction mixtures consisting of 25 μL (1 unit/well) of Jack bean (Canavalia ensiformis) urease, 55 μL of buffer at pH 6.8, 100 mM of urea, ...More data for this Ligand-Target Pair
Affinity DataKi: 2.15E+4nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Non-competitive inhibition of Saccharomyces cerevisiae alpha-glucosidase using p-nitrophenyl alpha-D-glucopyranoside as substrate preincubated for 15...More data for this Ligand-Target Pair
TargetOligo-1,6-glucosidase IMA1(Saccharomyces cerevisiae S288c (Baker's yeast))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 6.80E+4nMAssay Description:Competitive inhibition of Saccharomyces cerevisiae alpha-glucosidase using p-nitrophenyl alpha-D-glucopyranoside as substrate preincubated for 15 min...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 26.2nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured every 5 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured every 5 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In-vitro butyryl cholinesterase inhibitory activity was performed in 96-well microplates, 0.5 mM test compound in methanol, was incubated with 20 ...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human DNA topoisomerase 2beta after 2 hrs by ELISAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Fr£Res Mentouri-Constantine University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition measured every 5 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia
Curated by ChEMBL
Universiti Sains Malaysia
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair