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Found 29 with Last Name = 'wakil' and Initial = 'sj'
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM20182((1S,2R,5S,10S,11S,14R,15R)-14-[(2R)-6-hydroxy-6-me...)
Affinity DataIC50:  300nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  700nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351539(CHEMBL1824674)
Affinity DataIC50:  900nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351538(CHEMBL1824673)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351541(CHEMBL1824676)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351540(CHEMBL1824675)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351534(CHEMBL1824669)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351535(CHEMBL1824670)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351529(CHEMBL1824664)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351536(CHEMBL1824671)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351521(CHEMBL1824658)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351537(CHEMBL1824672)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351542(CHEMBL1824661)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351533(CHEMBL1824668)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351531(CHEMBL1824666)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351530(CHEMBL1824665)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351526(CHEMBL1616869)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM78179(2-(2-propyl-4-pyridyl)-4-(p-tolyl)thiazole;hydrobr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351528(CHEMBL1824663)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM93773(4-(4-chlorophenyl)-2-(2-propyl-4-pyridinyl)thiazol...)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351524(CHEMBL1824660)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351527(CHEMBL1824662)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351532(CHEMBL1824667)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351518(CHEMBL1824655)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351519(CHEMBL1824656)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351523(CHEMBL1824659)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351522(CHEMBL1300882 | cid_715106)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol regulatory element-binding protein 2(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50351520(CHEMBL1824657)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of SREBP2 activation expressed in CHO-K1 cells cotransfected with pSRE-Luc plasmid assessed as inhibition of luciferase expression after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed