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Found 75 with Last Name = 'wakimoto' and Initial = 't'
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  1.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  1.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  2.10nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  2.60nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40785(Calyculinamide A (18))
Affinity DataIC50:  5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  7.5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  8.20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40782(C1/C34-Calyculin A (15))
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  9nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40787(Des-N-methylcalyculin A (20))
Affinity DataIC50:  11nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40780(Calyculin A 21-acetate (13))
Affinity DataIC50:  13nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40777(Hemicalyculin A (5))
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  14nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  20nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40790(Calyculin C (24))
Affinity DataIC50:  29nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  55nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40781(Calyculin J (14))
Affinity DataIC50:  105nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  112nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40776(Calyculin A (4) | Calyculin B (19) | Calyculin E (...)
Affinity DataIC50:  185nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296237((2R,3R)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40784(Dephosphonocalyculin A (17))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40783(C9/C35-calyculin (16))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40779(Calyculin A 11,13,21-triacetate (12))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40778(11,13-O-isopropylidene-calyculin A (6))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40784(Dephosphonocalyculin A (17))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40783(C9/C35-calyculin (16))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40779(Calyculin A 11,13,21-triacetate (12))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein phosphatase 1 regulatory subunit 1A(Homo sapiens (Human))
The University Of Tokyo

LigandPNGBDBM40778(11,13-O-isopropylidene-calyculin A (6))
Affinity DataIC50: >1.00E+4nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296235((-)-Epigallocatechin-3-(4''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296236((2R,3R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296235((-)-Epigallocatechin-3-(4''-O-methyl)gallate | (2R...)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296234((-)-epigallocatechin-3-(3''-O-methyl)gallate | (2R...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296238((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296241((2R,3S)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296240((2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296239((2S,3R)-5,7-Dihydroxy-2-(3,4,5-trihydroxyphenyl)ch...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human recombinant MMP7 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296237((2R,3R)-2-(3,4-Dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human recombinant MMP2 expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Shizuoka And Global Coe Program

Curated by ChEMBL
LigandPNGBDBM50296240((2R,3S)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxychrom...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of human recombinant MT1-MMP expressed in Escherichia coli by fluorogenic peptide cleavage assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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