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Found 171 with Last Name = 'walpole' and Initial = 'cs'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052327(6-hydroxy-15-isopropenyl-4,13,17-trimethyl-5-oxo-(...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052320(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  1nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052323((4-Hydroxy-3-methoxy-phenyl)-acetic acid 4a,7b-dih...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052333(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052328(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052330(13-benzyl-5,6-dihydroxy-15-isopropenyl-4,17-dimeth...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052321(CHEMBL98634 | Phenyl-acetic acid (1aR,1bS,4aR,7aS,...)
Affinity DataKi:  600nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50052324(13-benzyl-6-hydroxy-8-hydroxymethyl-15-isopropenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataIC50:  2.90nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097740(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  410nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097732(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  510nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727((S)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50:  980nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733((S)-1-[N'-(2-Nitro-phenyl)-hydrazinothiocarbonyl]-...)
Affinity DataIC50:  1.67E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733((S)-1-[N'-(2-Nitro-phenyl)-hydrazinothiocarbonyl]-...)
Affinity DataIC50:  1.67E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097726(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097740(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733((S)-1-[N'-(2-Nitro-phenyl)-hydrazinothiocarbonyl]-...)
Affinity DataIC50:  2.31E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097730(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  2.43E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097742(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  3.60E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097743(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097738(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  4.50E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097725(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097731(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727((S)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50:  7.93E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727((S)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50:  7.93E+3nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097728(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097723(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  1.10E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097734(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  2.40E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097729(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  2.40E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097737(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  3.10E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097736(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50:  4.60E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727((S)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rabbit whole brain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724((R)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097731(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097738(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097726(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097742(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097724((R)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rabbit whole brain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097734(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097723(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097733((S)-1-[N'-(2-Nitro-phenyl)-hydrazinothiocarbonyl]-...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in rat whole forebrain membranes using [3H][Sar9Met(O2)]-SP binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097730(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097737(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097732(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097727((S)-1-{N'-[4-(2-Methylsulfanyl-ethylsulfamoyl)-2-n...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(RAT)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50097736(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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