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Found 19 with Last Name = 'watkins' and Initial = 'lr'
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089805(CHEMBL3577590)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089824(CHEMBL3577592)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089806(CHEMBL3577591)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089804(CHEMBL3576878)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089803(CHEMBL3577589)
Affinity DataIC50:  1.70E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089831(CHEMBL3577593)
Affinity DataIC50:  1.80E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089802(CHEMBL3577588)
Affinity DataIC50:  3.00E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089785(CHEMBL3577579)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089843(CHEMBL3577594)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089801(CHEMBL3577587)
Affinity DataIC50:  6.70E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089800(CHEMBL3577586)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089798(CHEMBL3577584)
Affinity DataIC50:  2.25E+4nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089799(CHEMBL3577585)
Affinity DataIC50:  2.48E+4nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089796(CHEMBL3577583)
Affinity DataIC50:  4.89E+4nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089784(CHEMBL3577578)
Affinity DataIC50:  7.62E+4nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089783(CHEMBL3577577)
Affinity DataIC50:  1.06E+5nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089795(CHEMBL3577582)
Affinity DataIC50:  1.18E+5nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089793(CHEMBL3577581)
Affinity DataIC50:  1.44E+5nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
National Institute Of Health

Curated by ChEMBL
LigandPNGBDBM50089792(CHEMBL3577580)
Affinity DataIC50:  2.43E+5nMAssay Description:Antagonist activity against TLR4 in mouse BV2 cells assessed as inhibition of LPS-induced nitric oxide production incubated for 24 hrs by 2,3-diamino...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed