Compile Data Set for Download or QSAR
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Found 32 with Last Name = 'welbourn' and Initial = 'ap'
LigandPNGBDBM50227383(CHEMBL556758)
Affinity DataKi:  0.160nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226939(CHEMBL36616)
Affinity DataKi:  0.240nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50227384(CHEMBL172132)
Affinity DataKi:  0.420nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226938(CHEMBL38829)
Affinity DataKi:  0.690nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226961(CHEMBL38788)
Affinity DataKi:  0.960nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226937(CHEMBL289153)
Affinity DataKi:  1.90nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50227384(CHEMBL172132)
Affinity DataKi:  1.90nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226964(CHEMBL41064)
Affinity DataKi:  3nMAssay Description:Inhibition of saturable binding of [3H]idazoxan to alpha2-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50226939(CHEMBL36616)
Affinity DataKi:  3.70nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50226961(CHEMBL38788)
Affinity DataKi:  3.70nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50226938(CHEMBL38829)
Affinity DataKi:  3.90nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50226964(CHEMBL41064)
Affinity DataKi:  8.40nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha1-site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50227383(CHEMBL556758)
Affinity DataKi:  13nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor site in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  16.3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50226937(CHEMBL289153)
Affinity DataKi:  18nMAssay Description:Inhibition of saturable binding of [3H]prazosin to alpha-1 adrenergic receptor in rat cerebral cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  256nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  449nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  449nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  487nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  8.73E+3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  8.73E+3nMAssay Description:Displacement of [3H]idazoxan from alpha-2 adrenergic receptor from rat brain cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225888(CHEMBL61325)
Affinity DataKi:  1.33E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  4.64E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Reckitt And Colman

Curated by ChEMBL
LigandPNGBDBM50225887(CHEMBL61234)
Affinity DataKi:  4.64E+4nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor from rat brain cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed