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Found 156 with Last Name = 'xie' and Initial = 'k'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86463((+)-6-fluorodinapsoline hydrobromide | CAS_0 | NSC...)
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117182(2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117181((S)-2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinol...)
Affinity DataKi:  11.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86454(6-ethyldinapsoline hydrobromide)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86178((+/-)-2-propyldinapsoline hydrobromide | Dinapsoli...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86456(4-hydroxydinapsoline hydrobromide)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86455((+/-)-11-chlorodinapsoline hydrobromide | CAS_0 | ...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86454(6-ethyldinapsoline hydrobromide)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86459(4-fluorodinapsoline hydrobromide | CAS_0 | NSC_0)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50309707(4-fluorobenzaldehyde O-4-butoxyphenylcarbamoyl oxi...)
Affinity DataKi:  30nMAssay Description:Competitive inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117181((S)-2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinol...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86461(1,2,3,11b-Tetrahydro[1]benzothiopyrano[4,3,2-de]is...)
Affinity DataKi:  34.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117181((S)-2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinol...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86462((+/-)-3-methyldinapsoline hydrobromide)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117182(2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-...)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117182(2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-...)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86459(4-fluorodinapsoline hydrobromide | CAS_0 | NSC_0)
Affinity DataKi:  69nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86466((+/-)-2-methyldinapsoline hydrobromide | CAS_0 | N...)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86456(4-hydroxydinapsoline hydrobromide)
Affinity DataKi:  72nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86470((+/-)-3-perfluorobutyldinapsoline hydrobromide | C...)
Affinity DataKi:  78nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86458((+/-)-3-n-butyldinapsoline hydrobromide)
Affinity DataKi:  93nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86465((+/-)-7-methyldinapsoline hydrobromide)
Affinity DataKi:  139nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86465((+/-)-7-methyldinapsoline hydrobromide)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86468(4-fluoro-2,3,7,11b-tetrahydro-1H-pyrido[3,4,5-k]ac...)
Affinity DataKi:  160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86464((-)-6-fluorodinapsoline hydrobromide | CAS_0 | NSC...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86458((+/-)-3-n-butyldinapsoline hydrobromide)
Affinity DataKi:  299nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86470((+/-)-3-perfluorobutyldinapsoline hydrobromide | C...)
Affinity DataKi:  340nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86466((+/-)-2-methyldinapsoline hydrobromide | CAS_0 | N...)
Affinity DataKi:  382nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86457((+/-)-7,7'-dimethyldinapsoline hydrobromide | ...)
Affinity DataKi:  390nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86460((+/-)-7-ethyldinapsoline hydrobromide)
Affinity DataKi:  430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86460((+/-)-7-ethyldinapsoline hydrobromide)
Affinity DataKi:  440nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86461(1,2,3,11b-Tetrahydro[1]benzothiopyrano[4,3,2-de]is...)
Affinity DataKi:  536nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86457((+/-)-7,7'-dimethyldinapsoline hydrobromide | ...)
Affinity DataKi:  870nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86471((+/-)-7-methoxycarbonylmethyldinapsoline)
Affinity DataKi:  990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86469((+/-)-11-nitrodinapsoline hydrobromide | CAS_0 | N...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86455((+/-)-11-chlorodinapsoline hydrobromide | CAS_0 | ...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117183(2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86462((+/-)-3-methyldinapsoline hydrobromide)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86178((+/-)-2-propyldinapsoline hydrobromide | Dinapsoli...)
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86471((+/-)-7-methoxycarbonylmethyldinapsoline)
Affinity DataKi:  2.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86464((-)-6-fluorodinapsoline hydrobromide | CAS_0 | NSC...)
Affinity DataKi:  3.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50117183(2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-...)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86467((+/-)-2,3-Dimethyldinapsoline hydrobromide | CAS_0...)
Affinity DataKi:  9.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86467((+/-)-2,3-Dimethyldinapsoline hydrobromide | CAS_0...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86469((+/-)-11-nitrodinapsoline hydrobromide | CAS_0 | N...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM86468(4-fluoro-2,3,7,11b-tetrahydro-1H-pyrido[3,4,5-k]ac...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50309725(CHEMBL598764 | nicotinaldehyde O-4-(undecyloxy)phe...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50309712(4-fluorobenzaldehyde O-4-(nonyloxy)phenylcarbamoyl...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50309701(CHEMBL597430 | benzaldehyde O-4-(nonyloxy)phenylca...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Bristol-Myers Squibb Research & Development

Curated by ChEMBL
LigandPNGBDBM50309713(4-fluorobenzaldehyde O-4-(decyloxy)phenylcarbamoyl...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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