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Found 60 with Last Name = 'xie' and Initial = 'n'
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384894(CHEMBL2036262)
Affinity DataIC50:  42.7nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  64.6nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384894(CHEMBL2036262)
Affinity DataIC50:  91.2nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096258(CHEMBL3593303)
Affinity DataIC50:  118nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096264(CHEMBL3593308)
Affinity DataIC50:  120nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384893(CHEMBL2036261)
Affinity DataIC50:  129nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096260(CHEMBL3593305)
Affinity DataIC50:  129nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096266(CHEMBL3593310)
Affinity DataIC50:  131nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096267(CHEMBL3593311)
Affinity DataIC50:  137nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096259(CHEMBL3593304)
Affinity DataIC50:  154nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384892(CHEMBL2036260)
Affinity DataIC50:  155nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096265(CHEMBL3593309)
Affinity DataIC50:  169nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096262(CHEMBL3593246)
Affinity DataIC50:  173nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384890(CHEMBL2036263)
Affinity DataIC50:  178nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384890(CHEMBL2036263)
Affinity DataIC50:  178nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096263(CHEMBL3593307)
Affinity DataIC50:  178nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384895(CHEMBL2036259)
Affinity DataIC50:  182nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50096261(CHEMBL3593306)
Affinity DataIC50:  217nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384891(CHEMBL2036258)
Affinity DataIC50:  229nMAssay Description:Inhibition of equine serum butyrylcholine esterase using butyrylcholine chloride as substrate incubated for 5 mins prior to substrate addition measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Academy Of Military Medical Sciences

Curated by ChEMBL
LigandPNGBDBM19410(CHEMBL27759 | MS-275 | US11377423, MS-275 | US1167...)
Affinity DataIC50:  273nMAssay Description:Inhibition of HDAC1 (unknown origin) preincubated for 5 mins followed by fluorogenic substrate addition measured after 30 mins by microplate reader a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  980nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384891(CHEMBL2036258)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255524(Ac-SGRGK(CoA)GGKGLGKGGAKRHRK | CHEMBL505605)
Affinity DataIC50:  2.88E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  4.35E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384895(CHEMBL2036259)
Affinity DataIC50:  6.03E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  6.62E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384892(CHEMBL2036260)
Affinity DataIC50:  7.24E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  7.54E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  8.15E+3nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50384893(CHEMBL2036261)
Affinity DataIC50:  8.32E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase using acetylcholine chloride as substrate incubated for 5 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50292429(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of TIP60 in human HeLa cell extracts by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  1.74E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  2.59E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50067040(((E,E)-1,7-bis(4-hydroxy-3-methoxyphenyl)-1,6-hept...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  4.19E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  4.59E+4nMAssay Description:Inhibition of recombinant p300More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255526(Ac-SGRGKGGKGLGK(CoA)GGAKRHRK | CHEMBL500256)
Affinity DataIC50:  5.36E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255527(Ac-SGRGKGGKGLGKGGAK(CoA)RHRK | CHEMBL504265)
Affinity DataIC50:  5.85E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255528(Ac-SGRGK(CoA)QGGKARAKAKTRSSRA | CHEMBL509144)
Affinity DataIC50:  6.05E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255524(Ac-SGRGK(CoA)GGKGLGKGGAKRHRK | CHEMBL505605)
Affinity DataIC50:  6.59E+4nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255522(Ac-ARTKQTARKSTGGK(CoA)APRKQL | CHEMBL526343)
Affinity DataIC50:  7.96E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50367033(COENZYME_A)
Affinity DataIC50:  8.23E+4nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  1.08E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  1.12E+5nMAssay Description:Inhibition of recombinant Tip60 (1-513) expressed in Escherichia coli BL21 (DE3) by liquid scintillationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50255525(Ac-SGRGKGGK(CoA)GLGKGGAKRHRK | CHEMBL448227)
Affinity DataIC50:  1.24E+5nMAssay Description:Inhibition of PCAF HAT domain (493-658) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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