Compile Data Set for Download or QSAR
maximum 50k data
Found 107 with Last Name = 'xing' and Initial = 'm'
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  100nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383835(CHEMBL2030993)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424979(CHEMBL2311747)
Affinity DataIC50:  180nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383830(CHEMBL2030988)
Affinity DataIC50:  220nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137968(CHEMBL3754002)
Affinity DataIC50:  280nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383816(CHEMBL2030974)
Affinity DataIC50:  420nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424976(CHEMBL2316785)
Affinity DataIC50:  460nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394508(CHEMBL2159921)
Affinity DataIC50:  500nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50:  570nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383836(CHEMBL2030978)
Affinity DataIC50:  650nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383825(CHEMBL2030983)
Affinity DataIC50:  780nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383834(CHEMBL2030992)
Affinity DataIC50:  790nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383829(CHEMBL2030987)
Affinity DataIC50:  840nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424980(CHEMBL2316794)
Affinity DataIC50:  850nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137968(CHEMBL3754002)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394505(CHEMBL2159925)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137851(CHEMBL3752866)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424977(CHEMBL2316784)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383815(CHEMBL2030973)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383820(CHEMBL1512579)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383824(CHEMBL2030982)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Mus musculus (Mouse))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137701(CHEMBL3752369)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of PI3K-gamma in mouse lymph node cells assessed as inhibition of ConA-stimulated T cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394500(CHEMBL2159924)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383831(CHEMBL2030989)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383826(CHEMBL2030984)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424978(CHEMBL2316777)
Affinity DataIC50:  2.23E+3nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383812(CHEMBL1533728)
Affinity DataIC50:  2.34E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50424981(CHEMBL2316793)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of human HER2 cytoplasmic domain (amino acids 676 to 1245) expressed in Sf9 cells by DELFIA time resolved fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383817(CHEMBL2030975)
Affinity DataIC50:  2.65E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394513(CHEMBL2160142)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394497(CHEMBL2160139)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383821(CHEMBL2030979)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394499(CHEMBL2159926)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383832(CHEMBL2030990)
Affinity DataIC50:  3.04E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50137701(CHEMBL3752369)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383827(CHEMBL2030985)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383813(CHEMBL2030971)
Affinity DataIC50:  3.57E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394501(CHEMBL2159923)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394506(CHEMBL2160146)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383818(CHEMBL2030976)
Affinity DataIC50:  4.79E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394498(CHEMBL2159927)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383833(CHEMBL2030991)
Affinity DataIC50:  5.52E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383822(CHEMBL2030980)
Affinity DataIC50:  5.59E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50383828(CHEMBL2030986)
Affinity DataIC50:  5.71E+3nMAssay Description:Inhibition of human recombinant Aurora A kinase using biotinylated peptide substrate preincubated for 15 mins with compound measured after 30 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394503(CHEMBL2160141)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394509(CHEMBL2159922)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Anhui Agricultural University

Curated by ChEMBL
LigandPNGBDBM50138037(CHEMBL3752051)
Affinity DataIC50:  6.57E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50394496(CHEMBL2158024)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of COX-2 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 107 total ) | Next | Last >>
Jump to: