Affinity DataKi: 0.800nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:In vitro binding affinity (agonistic) towards human CRTH2 receptor expressed in CHO cells; range 15 to 25 nMMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Mixed inhibition of hCES2A in human liver microsome assessed as reduction in fluorescein diacetate hydrolysis preincubated for 10 mins followed by su...More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
Affinity DataKi: 225nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
Affinity DataKi: 299nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 370nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) using Lys4-dimethylated H3 (1-20) peptide as substrate incubated for 30 mins by peroxidase-coupled ass...More data for this Ligand-Target Pair
Affinity DataKi: 457nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of recombinant human MAO-A expressed in Pichia pastoris using kynuramine as substrate by peroxidase-coupled methodMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) using Lys4-dimethylated H3 (1-20) peptide as substrate incubated for 30 mins by peroxidase-coupled ass...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 610nMAssay Description:Inhibition of hexahistidine-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli Rosetta (DE3) cells using H3K4me2 peptide as substr...More data for this Ligand-Target Pair
Affinity DataKi: 634nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 880nMAssay Description:Inhibition of human LSD1 (172 to 833 residues) using Lys4-dimethylated H3 (1-20) peptide as substrate incubated for 30 mins by peroxidase-coupled ass...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibitory activity against ALKMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human LSD1/CoREST expressed in Escherichia coli using histone H3 peptide monomethylated at Lys4 as substrate by peroxidase-coupled assa...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.15E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.17E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.18E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in Pichia pastoris using kynuramine as substrate by peroxidase-coupled methodMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.29E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of human LSD1/CoREST expressed in Escherichia coli using histone H3 peptide monomethylated at Lys4 as substrate by peroxidase-coupled assa...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.32E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.37E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetCocaine esterase(Homo sapiens (Human))
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of human CES2A using 4-methylumbelliferone as a substrateMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of LSD1 (unknown origin) using H3K4(diMe) peptide as substrate measured after 60 mins by amplex red dye based HRP-coupled assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of human LSD1/CoREST expressed in Escherichia coli using histone H3 peptide monomethylated at Lys4 as substrate by peroxidase-coupled assa...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 1.92E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 2.03E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in Pichia pastoris using kynuramine as substrate by peroxidase-coupled methodMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of hexahistidine-tagged human LSD1 (172 to 833 residues) expressed in Escherichia coli Rosetta (DE3) cells using H3K4me2 peptide as substr...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Institute For Life Science Research
Curated by ChEMBL
Institute For Life Science Research
Curated by ChEMBL
Affinity DataKi: 2.63E+3nMAssay Description:Binding affinity for human growth hormone secretagogue receptor was determined using [125I]-ghrelinMore data for this Ligand-Target Pair
Affinity DataKi: 2.98E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by peroxidase-coupled methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.86E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetInsulin receptor(Homo sapiens (Human))
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Chembridge Research Laboratories And Chembridge
Curated by ChEMBL
Affinity DataKi: 5.30E+3nMAssay Description:Inhibitory activity against IRKMore data for this Ligand-Target Pair
Affinity DataKi: 6.89E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Key Laboratory Of Henan Provinc
Curated by ChEMBL
Affinity DataKi: 7.40E+3nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by peroxidase-coupled methodMore data for this Ligand-Target Pair
Affinity DataKi: 7.71E+3nMAssay Description:Binding affinity towards human DP receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity towards human CRTH2 receptor expressed in CHO cells; range 25 nM to 8 uMMore data for this Ligand-Target Pair