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Found 92 with Last Name = 'yabannavar' and Initial = 'a'
LigandPNGBDBM50380236(CHEMBL2016856)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380229(CHEMBL2016996)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380230(CHEMBL2016862)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272192(4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(1...)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272242(6-(3-chlorophenyl)-4-(1H-indazol-5-yl)pyrimidin-2(...)
Affinity DataIC50:  5nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272244(6-(3-(benzyloxy)phenyl)-4-(1H-indazol-5-yl)pyrimid...)
Affinity DataIC50:  6nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380225(CHEMBL2017000)
Affinity DataIC50:  8nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380234(CHEMBL2016858)
Affinity DataIC50:  9nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272193(4-(1H-indazol-5-yl)-6-phenylpyrimidin-2(1H)-one | ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272240(6-(2-fluorophenyl)-4-(1H-indazol-5-yl)pyrimidin-2(...)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272191(4-(4-hydroxyphenyl)-6-phenylpyrimidin-2(1H)-one | ...)
Affinity DataIC50:  30nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380235(CHEMBL2016857)
Affinity DataIC50:  33nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380233(CHEMBL2016859)
Affinity DataIC50:  33nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272284(4-(1H-indazol-5-yl)-6-(4-(piperazin-1-yl)phenyl)py...)
Affinity DataIC50:  40nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380226(CHEMBL2016999)
Affinity DataIC50:  41nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272283(6-(4-ethylphenyl)-4-(1H-indazol-5-yl)pyrimidin-2(1...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272243(4-(1H-indazol-5-yl)-6-(3-(trifluoromethyl)phenyl)p...)
Affinity DataIC50:  110nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115465(2-(4-Allyloxy-3-trifluoromethoxy-phenyl)-4,5-dihyd...)
Affinity DataIC50:  120nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272241(6-(3-fluorophenyl)-4-(1H-indazol-5-yl)pyrimidin-2(...)
Affinity DataIC50:  150nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115478(2-(4-Methoxy-3-trifluoromethoxy-phenyl)-4,5-dihydr...)
Affinity DataIC50:  160nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115438(2-[4-(3-Methyl-but-2-enyloxy)-3-trifluoromethoxy-p...)
Affinity DataIC50:  190nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115468(2-[4-(3-Fluoro-benzyloxy)-3-trifluoromethoxy-pheny...)
Affinity DataIC50:  250nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115464(2-(4'-Propyl-biphenyl-4-yl)-4,5-dihydro-oxazole-4-...)
Affinity DataIC50:  280nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115437(2-(3-Chloro-5-fluoro-1H-indol-2-yl)-4,5-dihydro-ox...)
Affinity DataIC50:  300nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115430(2-(4-But-3-enyloxy-3-trifluoromethoxy-phenyl)-4,5-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272282(6-(4-(benzyloxy)phenyl)-4-(1H-indazol-5-yl)pyrimid...)
Affinity DataIC50:  350nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380232(CHEMBL2016860)
Affinity DataIC50:  370nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115457(2-(4-Methoxy-3-propyl-5-trifluoromethoxy-phenyl)-4...)
Affinity DataIC50:  500nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115426(2-[4-(3-Nitro-phenoxymethyl)-phenyl]-4,5-dihydro-o...)
Affinity DataIC50:  560nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115471(2-[3-Fluoro-4-(3-trifluoromethyl-benzyloxy)-phenyl...)
Affinity DataIC50:  840nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115443(2-(4-Fluoro-3-propyl-phenyl)-4,5-dihydro-oxazole-4...)
Affinity DataIC50:  960nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Novartis Institutes Of Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50272286(4-(2-aminopyridin-4-yl)-6-(2,4-dimethoxyphenyl)pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of CDC7-DBF4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115477(2-(3-Ethoxy-4-fluoro-phenyl)-4,5-dihydro-oxazole-4...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115455(2-[4-(3-Nitro-benzyloxy)-phenyl]-4,5-dihydro-oxazo...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115436(2-(4-Fluoro-3-methyl-phenyl)-4,5-dihydro-oxazole-4...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115470(2-(4-Fluoro-3-trifluoromethyl-phenyl)-4,5-dihydro-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115472(2-(4-Allyloxy-3-fluoro-phenyl)-4,5-dihydro-oxazole...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115460(4-(1,1-Difluoro-ethoxy)-N-(2-hydroxy-1-hydroxycarb...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115463(2-(5-Fluoro-1H-indol-2-yl)-4,5-dihydro-oxazole-4-c...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115435(2-(4-Allyloxy-3-trifluoromethyl-phenyl)-4,5-dihydr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115431(2-(3-Trifluoromethyl-phenyl)-4,5-dihydro-oxazole-4...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115439(2-(4-Bromo-phenyl)-4,5-dihydro-oxazole-4-carboxyli...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115474(2-(3-Allyl-5-fluoro-4-methoxy-2-methyl-phenyl)-4,5...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115447(4-But-3-enyloxy-N-(2-hydroxy-1-hydroxycarbamoyl-et...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115444(2-(3-Bromo-4-fluoro-phenyl)-4,5-dihydro-oxazole-4-...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115427(2-(4-Dimethylamino-phenyl)-4,5-dihydro-oxazole-4-c...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115484(2-(4-Trifluoromethoxy-phenyl)-4,5-dihydro-oxazole-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50380238(CHEMBL2017001)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of CDC7/DBF4 using MCM-2 as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115442(2-(4-Nitro-phenyl)-4,5-dihydro-oxazole-4-carboxyli...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Chiron

Curated by ChEMBL
LigandPNGBDBM50115461(2-(4-Iodo-phenyl)-4,5-dihydro-oxazole-4-carboxylic...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of P. aeruginosa UDP-3-O-acyl-N-acetylglucosamine Deacetylase (LpxC) in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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