TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Tokushima Research Institute
Curated by PDSP Ki Database
Tokushima Research Institute
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Tokushima Research Institute
Curated by PDSP Ki Database
Tokushima Research Institute
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Tokushima Research Institute
Curated by PDSP Ki Database
Tokushima Research Institute
Curated by PDSP Ki Database
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.02E+3nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Suntory Institute For Bioorganic Research
Curated by PDSP Ki Database
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant DPP-8 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of human recombinant DPP-8 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant DPP-8 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of human recombinant DPP-8 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair