Affinity DataKi: 0.700nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.940nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 17nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 35nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 75nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 130nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 530nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(GUINEA PIG)
Syntex Discovery Research
Curated by PDSP Ki Database
Syntex Discovery Research
Curated by PDSP Ki Database
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.70E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.03E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human EP1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Inhibition of JAK3 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of JAK3 (unknown origin) using [33gammaP]ATP and Biotin-KAIETDKEYYTVKD as substrate incubated for 10 mins prior to substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of JAK3 (unknown origin) using [33gammaP]ATP and Biotin-KAIETDKEYYTVKD as substrate incubated for 10 mins prior to substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of JAK3 (unknown origin) using [33gammaP]ATP and Biotin-KAIETDKEYYTVKD as substrate incubated for 10 mins prior to substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of JAK3 (unknown origin) using [33gammaP]ATP and Biotin-KAIETDKEYYTVKD as substrate incubated for 10 mins prior to substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibition of JAK3 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Inhibition of JAK1 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK2 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 0.590nMAssay Description:Inhibition of JAK1 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK3 (unknown origin) using [33gammaP]ATP and Biotin-KAIETDKEYYTVKD as substrate incubated for 10 mins prior to substrate addition meas...More data for this Ligand-Target Pair
Affinity DataIC50: 0.741nMAssay Description:The chromogenic substrate D-Pro-Phe-Arg-pNa, 2HCl (BIOPHEN CS-31(02) from Hyphen BioMed, Neuville-Sur-oise, France) was dissolved in 5 mL deionized w...More data for this Ligand-Target Pair