Affinity DataKi: 0.0400nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.114nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
Affinity DataKi: 0.115nMAssay Description:Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.125nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:pA2 is the negative log of the molar concentration required to double the agonism of opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for Opioid receptor delta 1 using [3H]-DPDPE in rat brain P2 synaptosomal preparationMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Compound was tested for binding affinity towards opioid receptor delta 1 by displacing [3H]DPDPE radioligand in rat brain P2 synaptosomes membranes.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
National Institutes Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair