TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 9 (ADAM9)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 5.93nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 7.40nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 7.5nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 17 (ADAM17, TACE)More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 10 (ADAM10)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of CDK1/cyclin B after 40 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 16.7nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 24.8nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity at recombinant human histamine H4 receptor expressed in CHO-K1 cells assessed as inhibition of R-alpha-methylhistamine induced st...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Bos taurus)
Chong Kun Dang Research Institute
Curated by ChEMBL
Chong Kun Dang Research Institute
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of bovine PDE5More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 40.5nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Department Of Life Science And National Research Laboratory Of Proteolysis
Curated by ChEMBL
Affinity DataIC50: 42.3nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]BRL 43694 from human recombinant 5-HT3 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Institute Of Science And Technology
Curated by ChEMBL
Institute Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair