TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of rat Nav1.4 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of rat Nav1.3 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of rat Nav1.2 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
Affinity DataIC50: 3.96E+4nMAssay Description:Inhibition of mouse Nav1.6 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by t...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 5.23E+4nMAssay Description:Inhibition of rat Nav1.2 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 5.43E+4nMAssay Description:Inhibition of rat Nav1.4 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
Affinity DataIC50: 5.43E+4nMAssay Description:Inhibition of mouse Nav1.6 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by t...More data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of rat Nav1.3 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.74E+5nMAssay Description:Inhibition of rat Nav1.1 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.77E+5nMAssay Description:Inhibition of rat Nav1.7 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.04E+5nMAssay Description:Inhibition of rat Nav1.4 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 2.87E+5nMAssay Description:Inhibition of rat Nav1.5 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.3 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.7 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat Nav1.1 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 8.71E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 5.30nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 55nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Inhibition of rat Nav1.7 channel expressed in Xenopus oocyte by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Rattus norvegicus (Rat))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 50nMAssay Description:Inhibition of rat Nav1.4 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Rattus norvegicus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Inhibition of rat Nav1.3 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Binding affinity to rat voltage-gated sodium channel Nav1.2 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSodium channel protein type 1 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 290nMAssay Description:Inhibition of rat Nav1.1 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Inhibition of rat Nav1.2 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair