TargetKappa-type opioid receptor(Homo sapiens (Human))
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H]diprenorphine from human cloned kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]diprenorphine from human cloned mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-40 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity to amyloid beta aggregates in postmortem human Alzheimer's disease brain homogenates after 2 hrs by gamma countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-42 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-40) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Biomedizinische Forschungsreagenzien
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-42) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-40) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-42 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]Pittsburgh compound B from human Abeta1-40 after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Technische Universit£T M£Nchen
Curated by ChEMBL
Technische Universit£T M£Nchen
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]PiB from human amyloid beta (1-42) at 100 nM after 180 mins by liquid scintillation counterMore data for this Ligand-Target Pair