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Found 170 with Last Name = 'yuan' and Initial = 'l'
TargetChitin synthase 1(Candida albicans)
Shaanxi University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50559071(CHEMBL4741395)
Affinity DataKi:  0.550nMAssay Description:Inhibition of Candida albicans chitin synthase 1 expressed in Saccharomyces cerevisiae RRA400-1U cells using [3H]UDP-GlcNAc as substrate by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602006(CHEMBL5209436)
Affinity DataKi:  65nMAssay Description:Mixed type inhibition of Helicobacter pyroli urease assessed as dissociation constant for EI complex by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetChitin synthase 1(Candida albicans)
Shaanxi University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50559072(CHEMBL4786444)
Affinity DataKi:  630nMAssay Description:Inhibition of Candida albicans chitin synthase 1 expressed in Saccharomyces cerevisiae RRA400-1U cells using [3H]UDP-GlcNAc as substrate by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602006(CHEMBL5209436)
Affinity DataKi:  1.20E+3nMAssay Description:Mixed type inhibition of Helicobacter pyroli urease assessed as dissociation constant for ESI complex by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59188(Dihydroisoxazole, 3e)
Affinity DataKi:  4.30E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59187(Dihydroisoxazole, 3d)
Affinity DataKi:  6.10E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59186(Dihydroisoxazole, 3c)
Affinity DataKi:  7.80E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59190(Dihydroisoxazole, 4)
Affinity DataKi:  7.90E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59185(Dihydroisoxazole, 3b)
Affinity DataKi:  8.10E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59189(Dihydroisoxazole, 3f)
Affinity DataKi:  8.70E+4nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59177(Dihydroisoxazole, 1e | Dihydroisoxazole, 1f)
Affinity DataKi:  1.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59179(Dihydroisoxazole, 1g)
Affinity DataKi:  2.40E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59183(Dihydroisoxazole, 2b)
Affinity DataKi:  2.60E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59180(Dihydroisoxazole, 1h)
Affinity DataKi:  3.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59177(Dihydroisoxazole, 1e | Dihydroisoxazole, 1f)
Affinity DataKi:  3.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59176(Dihydroisoxazole, 1d)
Affinity DataKi:  3.90E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59174(Dihydroisoxazole, 1b)
Affinity DataKi:  4.20E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59175(Dihydroisoxazole, 1c)
Affinity DataKi:  4.30E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59173(Dihydroisoxazole, 1a)
Affinity DataKi:  7.40E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59181(Dihydroisoxazole, 1i)
Affinity DataKi:  9.10E+5nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59182(Dihydroisoxazole, 2a)
Affinity DataKi:  1.30E+6nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Stanford University

LigandPNGBDBM59184(Dihydroisoxazole, 3a)
Affinity DataKi:  2.70E+6nMpH: 7.2Assay Description:Recombinant of human TG2 was expressed in E.coli and purified to >90% homogeneity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of fluormone VDR red from human full-length VDR after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetEndochitinase B1(Aspergillus fumigatus)
Shaanxi University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50559069(CHEMBL4756641)
Affinity DataIC50:  27nMAssay Description:Inhibition of Aspergillus fumigatus chitinase B1 expressed in Escherichia coli using 4MU-GlcNAc2 as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetStimulator of interferon genes protein(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50605474(CHEMBL5189857)
Affinity DataIC50:  76nMAssay Description:Inhibition of STING (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50469127(CHEMBL4288947)
Affinity DataIC50:  89nMAssay Description:Displacement of fluormone VDR red from human full-length VDR after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50126186(2-(3-Naphthalen-2-yl-but-2-enoylamino)-benzoic aci...)
Affinity DataIC50:  93nMAssay Description:Inhibition of human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50441900(CHEMBL2434990)
Affinity DataIC50:  115nMAssay Description:Displacement of fluormone VDR red from human full-length VDR after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50469128(CHEMBL4290851)
Affinity DataIC50:  125nMAssay Description:Displacement of fluormone VDR red from human full-length VDR after 4 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602006(CHEMBL5209436)
Affinity DataIC50:  130nMAssay Description:Inhibition of Helicobacter pylori ureaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274307(CHEMBL511111 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  230nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274303(CHEMBL502862 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  240nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274292(CHEMBL509768 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  400nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274300(CHEMBL509633 | p-Methoxyphenyl (9-(4-biphenyl)meth...)
Affinity DataIC50:  470nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50446421(CHEMBL3109740)
Affinity DataIC50:  470nMAssay Description:Inhibition of human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50469128(CHEMBL4290851)
Affinity DataIC50:  650nMAssay Description:Binding affinity to VDR in scrambled siRNA-transfected human MCF7 cells assessed as cell growth inhibition by measuring reduction in BrdU incorporati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602003(CHEMBL5207136)
Affinity DataIC50:  740nMAssay Description:Inhibition of Helicobacter pylori ureaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274296(CHEMBL501599 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  900nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50469127(CHEMBL4288947)
Affinity DataIC50:  970nMAssay Description:Binding affinity to VDR in scrambled siRNA-transfected human MCF7 cells assessed as cell growth inhibition by measuring reduction in BrdU incorporati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50160391(CHEMBL3786231)
Affinity DataIC50:  980nMAssay Description:Inhibition of telomerase in human MGC-803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274291(CHEMBL502788 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274289(CHEMBL503830 | p-Methoxyphenyl (9-(4-biphenylcarbo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50160320(CHEMBL3786261)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of telomerase in human MGC-803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274306(CHEMBL505326 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  1.73E+3nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602005(CHEMBL5188176)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of Helicobacter pylori ureaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetB-cell receptor CD22(Homo sapiens (Human))
Gifu University

Curated by ChEMBL
LigandPNGBDBM50274308(CHEMBL504222 | p-Methoxyphenyl (3,5,9-trideoxy-5-g...)
Affinity DataIC50:  1.76E+3nMAssay Description:Binding affinity to biotinylated human CD22-human IgG1 chimeric protein expressed in mouse J558LST6 cells by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50160330(CHEMBL3785281)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of telomerase in human MGC-803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50160326(CHEMBL3787380)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of telomerase in human MGC-803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50160312(CHEMBL3786734)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of telomerase in human MGC-803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease subunit beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
National Demonstration Center For Experimental Chemistry Education

Curated by ChEMBL
LigandPNGBDBM50602012(CHEMBL5209403)
Affinity DataIC50:  2.41E+3nMAssay Description:Inhibition of Helicobacter pylori ureaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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