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Found 26 with Last Name = 'zahn' and Initial = 'tj'
LigandPNGBDBM50090637((2Z,6E)-7,11-dimethyl-3-(prop-1-en-2-yl)dodeca-2,6...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081229(10-(tert-butyl)-2,6-dimethyl-(6E,10Z)-2,6,10-dodec...)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081229(10-(tert-butyl)-2,6-dimethyl-(6E,10Z)-2,6,10-dodec...)
Affinity DataIC50:  31nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090639((2Z,6E)-7,11-dimethyl-3-(propan-2-yl)dodeca-2,6,10...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50100979(Phosphoric acid di-((2Z,6E,10E)-3,7,11,15-tetramet...)
Affinity DataIC50:  100nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090636((2Z,6E)-3-(butan-2-yl)-7,11-dimethyldodeca-2,6,10-...)
Affinity DataIC50:  102nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081235(3-substituted farnesyl diphosphate analogue | 4-[(...)
Affinity DataIC50:  119nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081234(3-[(Z)-ethylidene]-7,11-dimethyl-(6E)-1,6,10-dodec...)
Affinity DataIC50:  173nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081234(3-[(Z)-ethylidene]-7,11-dimethyl-(6E)-1,6,10-dodec...)
Affinity DataIC50:  173nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081235(3-substituted farnesyl diphosphate analogue | 4-[(...)
Affinity DataIC50:  189nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081227(10-ethyl-2,6-dimethyl-(6E,10E)-2,6,10-dodecatriene...)
Affinity DataIC50:  215nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090642((2Z,6E)-7,11-dimethyl-3-(2-methylpropyl)dodeca-2,6...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081226(1-[1-[(Z)-ethylidene]-5,9-dimethyl-(4E)-4,8-decadi...)
Affinity DataIC50:  299nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50100978(Phosphoric acid di-((2E,6Z,10E)-3,7,11,15-tetramet...)
Affinity DataIC50:  340nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081238(4-[(Z)-ethylidene]-8,12,16-trimethyl-(7E,11E)-1,7,...)
Affinity DataIC50:  453nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090638((2E,6E)-7,11-dimethyl-3-propyldodeca-2,6,10-trien-...)
Affinity DataIC50:  453nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081233(3-[(Z)-ethylidene]-7,11,15-trimethyl-(6E,10E)-1,6,...)
Affinity DataIC50:  715nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081233(3-[(Z)-ethylidene]-7,11,15-trimethyl-(6E,10E)-1,6,...)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081238(4-[(Z)-ethylidene]-8,12,16-trimethyl-(7E,11E)-1,7,...)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090641((2Z,6E)-3-(2,2-dimethylpropyl)-7,11-dimethyldodeca...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50090640(3-substituted farnesyl diphosphate analogue | {[(2...)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibitory activity against recombinant mammalian protein Farnesyltransferase expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081229(10-(tert-butyl)-2,6-dimethyl-(6E,10Z)-2,6,10-dodec...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081235(3-substituted farnesyl diphosphate analogue | 4-[(...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081234(3-[(Z)-ethylidene]-7,11-dimethyl-(6E)-1,6,10-dodec...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081227(10-ethyl-2,6-dimethyl-(6E,10E)-2,6,10-dodecatriene...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081226(1-[1-[(Z)-ethylidene]-5,9-dimethyl-(4E)-4,8-decadi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed