TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 2.70E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 3.20E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 5.80E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 7.10E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 5.30E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 5.30E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 3.40E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 1.50E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 5.70E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 1.40E+4nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 8.50E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini
Curated by ChEMBL
Istituto Giannina Gaslini
Curated by ChEMBL
Affinity DataEC50: 9.50E+3nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair