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Found 1411 with Last Name = 'zhao' and Initial = 'm'
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.0636nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50029085(CHEBI:83405 | CHEMBL525191 | GDC-0879)
Affinity DataKi:  0.130nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.143nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86416(Dmt-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  0.145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.151nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85736(Dmt-d-Arg-Phe-Orn-NH2 | H-Dmt-D-Arg-Phe-Orn-NH2)
Affinity DataKi:  0.161nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.163nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  0.172nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.173nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86418(Dmt-d-Ala-Phe-Phe-NH2)
Affinity DataKi:  0.174nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | Morphine | NSC_5980)
TargetMu-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  1.18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86417(5-amino-2-{1-[1-[1-amino-2-(4-hydroxyphenyl)ethylc...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  1.22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM50060070((S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phe...)
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86419(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266505(CHEMBL515526 | N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM26237(CHEMBL458242 | N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86415(Tyr-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  2.55nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266476(CHEMBL508786 | N-[6-((R)-2-Methoxymethylpyrrolidin...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86253(CAS_100929-53-1 | DAMGO | NSC_104742 | US10836728,...)
Affinity DataKi:  2.83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM50060070((S)-2-Amino-N-{(R)-1-[(S)-1-((S)-1-carbamoyl-2-phe...)
Affinity DataKi:  3.44nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266384(CHEMBL456287 | N-[6-(3,4-Dihydro-1H-isoquinolin-2-...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM85731([Dmt1]DALDA)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266416(CHEMBL458224 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1B1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50432672(CHEMBL2347912)
Affinity DataKi:  5.60nMAssay Description:Inhibition of human microsomal CYP1B1-dependent ethoxyresorufin-O-deethylase activity by spectrofluorimetric analysis in presence of NADPH regenerati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | Morphine | NSC_5980)
Affinity DataKi:  5.64nMMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50255246(CHEMBL469488 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266474(CHEMBL455848 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266415(CHEMBL516168 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86417(5-amino-2-{1-[1-[1-amino-2-(4-hydroxyphenyl)ethylc...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266476(CHEMBL508786 | N-[6-((R)-2-Methoxymethylpyrrolidin...)
Affinity DataKi:  10.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266381(CHEMBL515992 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86415(Tyr-d-Arg-Phe-A2pr-NH2)
Affinity DataKi:  12.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Cornell University

Curated by PDSP Ki Database
LigandPNGBDBM86419(CAS_122222 | DALDA | NSC_122222)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50432672(CHEMBL2347912)
Affinity DataKi:  14nMAssay Description:Inhibition of human microsomal CYP1A2-dependent methoxyresorufin-O-demethylase activity by spectrofluorimetric analysis in presence of NADPH regenera...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266504(CHEMBL456069 | N-[6-((S)-2-Methoxymethylpyrrolidin...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1B1(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataKi:  16nMAssay Description:Inhibition of human microsomal CYP1B1-dependent ethoxyresorufin-O-deethylase activity by spectrofluorimetric analysis in presence of NADPH regenerati...More data for this Ligand-Target Pair
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50229128(CHEMBL401401 | N-((S)-1-oxo-1-((S)-5-phenyl-1-(phe...)
Affinity DataKi:  19nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50255188(CHEMBL480444 | [2-(3,5-Dimethylpyrazol-1-yl)-6-((R...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266416(CHEMBL458224 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  19nMAssay Description:Inhibition of human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50255185(CHEMBL480443 | N-[6-((R)-2-Methoxymethylpyrrolidin...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataKi:  20nMAssay Description:Inhibition of human microsomal CYP1A2-dependent methoxyresorufin-O-demethylase activity by spectrofluorimetric analysis in presence of NADPH regenera...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens)
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50553786(CHEMBL4789106)
Affinity DataKi:  22nMAssay Description:Reversible inhibition of wild-type human SHP2 using DiFMUP as substrate and measured by jump dilution assayMore data for this Ligand-Target Pair
Target InfoPDB
GoogleScholar
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266475(CHEMBL455849 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266441(CHEMBL515344 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  25.8nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266412(CHEMBL456051 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266503(CHEMBL456068 | N-[6-((S)-2-Methoxymethylpyrrolidin...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50266385(CHEMBL456073 | N-[2-(3,5-Dimethylpyrazol-1-yl)-6-(...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Xavier University Of Louisiana

Curated by ChEMBL
LigandPNGBDBM50113259(CHEMBL3601433)
Affinity DataKi:  30nMAssay Description:Inhibition of human microsomal CYP1A2-dependent methoxyresorufin-O-demethylase activity by spectrofluorimetric analysis in presence of NADPH regenera...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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