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16 similar compounds to monomer 50232160

Compile data set for download or QSAR
Wt: 352.3
BDBM50232172
Wt: 316.3
BDBM50232173
Wt: 401.2
BDBM50232176
Wt: 317.3
BDBM50232161
Wt: 476.5
BDBM50232210
Wt: 461.8
BDBM50232162
Wt: 395.4
BDBM50232165
Wt: 332.3
BDBM50232166
Wt: 317.3
BDBM50232168
Wt: 334.3
BDBM50232170
Wt: 480.9
BDBM50232213
Wt: 480.9
BDBM50232205
Wt: 806.7
BDBM50232196
Wt: 834.7
BDBM50232198
Wt: 848.8
BDBM50232208
Displayed 1 to 15 (of 16 total )  |  Next  |  Last  >>

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 24 hits for monomerid = 50232172,50232173,50232176,50232161,50232210,50232162,50232165,50232166,50232168,50232170,50232213,50232205,50232196,50232198,50232208   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Estrogen-related receptor alpha


(Homo sapiens (Human))
BDBM50232196
PNG
(CHEMBL4102983)
Show SMILES C[C@@H]1CN(CCN1c1ccc(cn1)C(C)=O)C(=O)c1cc2c(C)nn(Cc3cccc(OCCNC(=O)CCC4=[N+]5C(C=C4)=Cc4c(C)cc(C)n4[B-]5(F)F)c3)c2s1
Show InChI InChI=1S/C42H45BF2N8O4S/c1-26-19-27(2)52-37(26)21-34-11-10-33(53(34)43(52,44)45)12-14-40(55)46-15-18-57-35-8-6-7-31(20-35)25-51-42-36(29(4)48-51)22-38(58-42)41(56)49-16-17-50(28(3)24-49)39-13-9-32(23-47-39)30(5)54/h6-11,13,19-23,28H,12,14-18,24-25H2,1-5H3,(H,46,55)/t28-/m1/s1
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n/an/a 650n/an/an/an/an/an/a



Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL


Assay Description
Inverse agonist activity at GAL4-fused human ERRalpha expressed in HEK293 cells assessed as inhibition of transcriptional activity after 20 hrs by lu...


Bioorg Med Chem Lett 27: 1145-1148 (2017)


Article DOI: 10.1016/j.bmcl.2017.01.076
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM50232213
PNG
(CHEMBL4069460)
Show SMILES CCCc1nc2ccc(cc2n1Cc1ccc(cc1)-c1ccccc1C(O)=O)-c1ccccc1Cl
Show InChI InChI=1S/C30H25ClN2O2/c1-2-7-29-32-27-17-16-22(24-9-5-6-11-26(24)31)18-28(27)33(29)19-20-12-14-21(15-13-20)23-8-3-4-10-25(23)30(34)35/h3-6,8-18H,2,7,19H2,1H3,(H,34,35)
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n/an/an/an/a 1.39E+3n/an/an/an/a



University of Innsbruck

Curated by ChEMBL


Assay Description
Transactivation of Gal4 fused human PPARgamma LBD expressed in African green monkey COS7 cells after 42 hrs by dual luciferase reporter gene assay


Eur J Med Chem 126: 590-603 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.051
More data for this
Ligand-Target Pair
Estrogen-related receptor alpha


(Homo sapiens (Human))
BDBM50232208
PNG
(CHEMBL4067818)
Show SMILES C[C@@H]1CN(CCN1c1ccc(cn1)C(C)=O)C(=O)c1cc2c(C)nn(Cc3cccc(OCCCCCNC(=O)CCC4=[N+]5C(C=C4)=Cc4c(C)cc(C)n4[B-]5(F)F)c3)c2s1
Show InChI InChI=1S/C45H51BF2N8O4S/c1-29-22-30(2)55-40(29)24-37-14-13-36(56(37)46(55,47)48)15-17-43(58)49-18-7-6-8-21-60-38-11-9-10-34(23-38)28-54-45-39(32(4)51-54)25-41(61-45)44(59)52-19-20-53(31(3)27-52)42-16-12-35(26-50-42)33(5)57/h9-14,16,22-26,31H,6-8,15,17-21,27-28H2,1-5H3,(H,49,58)/t31-/m1/s1
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n/an/a 80n/an/an/an/an/an/a



Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL


Assay Description
Inverse agonist activity at GAL4-fused human ERRalpha expressed in HEK293 cells assessed as inhibition of transcriptional activity after 20 hrs by lu...


Bioorg Med Chem Lett 27: 1145-1148 (2017)


Article DOI: 10.1016/j.bmcl.2017.01.076
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232161
PNG
(CHEMBL4091622)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccncc2)c1F
Show InChI InChI=1S/C16H9F2NO2S/c17-10-1-2-11(20)15(18)14(10)16(21)13-4-3-12(22-13)9-5-7-19-8-6-9/h1-8,20H
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n/an/a 150n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232168
PNG
(CHEMBL4101849)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2cccnc2)c1F
Show InChI InChI=1S/C16H9F2NO2S/c17-10-3-4-11(20)15(18)14(10)16(21)13-6-5-12(22-13)9-2-1-7-19-8-9/h1-8,20H
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n/an/a 47n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232162
PNG
(CHEMBL4082298)
Show SMILES COc1c(Cl)cc(cc1Cn1ccnn1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C21H14ClF2N3O3S/c1-30-21-12(10-27-7-6-25-26-27)8-11(9-13(21)22)16-4-5-17(31-16)20(29)18-14(23)2-3-15(28)19(18)24/h2-9,28H,10H2,1H3
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n/an/a 9n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232166
PNG
(CHEMBL4071588)
Show SMILES Oc1ccc(cc1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C17H10F2O3S/c18-11-5-6-12(21)16(19)15(11)17(22)14-8-7-13(23-14)9-1-3-10(20)4-2-9/h1-8,20-21H
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n/an/a 3n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232170
PNG
(CHEMBL4071808)
Show SMILES Oc1cccc(C(=O)c2ccc(s2)-c2ccc(F)cc2F)c1F
Show InChI InChI=1S/C17H9F3O2S/c18-9-4-5-10(12(19)8-9)14-6-7-15(23-14)17(22)11-2-1-3-13(21)16(11)20/h1-8,21H
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n/an/a 47n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232173
PNG
(CHEMBL4083849)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccccc2)c1F
Show InChI InChI=1S/C17H10F2O2S/c18-11-6-7-12(20)16(19)15(11)17(21)14-9-8-13(22-14)10-4-2-1-3-5-10/h1-9,20H
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n/an/a 35n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232172
PNG
(CHEMBL4080385)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccc(F)cc2F)c1F
Show InChI InChI=1S/C17H8F4O2S/c18-8-1-2-9(11(20)7-8)13-5-6-14(24-13)17(23)15-10(19)3-4-12(22)16(15)21/h1-7,22H
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n/an/a 9n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232165
PNG
(CHEMBL4067584)
Show SMILES NS(=O)(=O)c1cccc(c1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C17H11F2NO4S2/c18-11-4-5-12(21)16(19)15(11)17(22)14-7-6-13(25-14)9-2-1-3-10(8-9)26(20,23)24/h1-8,21H,(H2,20,23,24)
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n/an/a 86n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232161
PNG
(CHEMBL4091622)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccncc2)c1F
Show InChI InChI=1S/C16H9F2NO2S/c17-10-1-2-11(20)15(18)14(10)16(21)13-4-3-12(22-13)9-5-7-19-8-6-9/h1-8,20H
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n/an/a 39n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232162
PNG
(CHEMBL4082298)
Show SMILES COc1c(Cl)cc(cc1Cn1ccnn1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C21H14ClF2N3O3S/c1-30-21-12(10-27-7-6-25-26-27)8-11(9-13(21)22)16-4-5-17(31-16)20(29)18-14(23)2-3-15(28)19(18)24/h2-9,28H,10H2,1H3
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n/an/a 2.10n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232166
PNG
(CHEMBL4071588)
Show SMILES Oc1ccc(cc1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C17H10F2O3S/c18-11-5-6-12(21)16(19)15(11)17(22)14-8-7-13(23-14)9-1-3-10(20)4-2-9/h1-8,20-21H
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n/an/a 71n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232176
PNG
(CHEMBL4091749)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2cc(Cl)c(O)c(Cl)c2)c1F
Show InChI InChI=1S/C17H8Cl2F2O3S/c18-8-5-7(6-9(19)16(8)23)12-3-4-13(25-12)17(24)14-10(20)1-2-11(22)15(14)21/h1-6,22-23H
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n/an/a 39n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232168
PNG
(CHEMBL4101849)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2cccnc2)c1F
Show InChI InChI=1S/C16H9F2NO2S/c17-10-3-4-11(20)15(18)14(10)16(21)13-6-5-12(22-13)9-2-1-7-19-8-9/h1-8,20H
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n/an/a 27n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232173
PNG
(CHEMBL4083849)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccccc2)c1F
Show InChI InChI=1S/C17H10F2O2S/c18-11-6-7-12(20)16(19)15(11)17(21)14-9-8-13(22-14)10-4-2-1-3-5-10/h1-9,20H
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n/an/a 11n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232172
PNG
(CHEMBL4080385)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2ccc(F)cc2F)c1F
Show InChI InChI=1S/C17H8F4O2S/c18-8-1-2-9(11(20)7-8)13-5-6-14(24-13)17(23)15-10(19)3-4-12(22)16(15)21/h1-7,22H
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n/an/a 3.5n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 2


(Homo sapiens (Human))
BDBM50232170
PNG
(CHEMBL4071808)
Show SMILES Oc1cccc(C(=O)c2ccc(s2)-c2ccc(F)cc2F)c1F
Show InChI InChI=1S/C17H9F3O2S/c18-9-4-5-10(12(19)8-9)14-6-7-15(23-14)17(22)11-2-1-3-13(21)16(11)20/h1-8,21H
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n/an/a 55n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental microsomal 17beta-HSD2 using [2,4,6,7-3H]-E2 as substrate after 20 mins in presence of NAD+ by RP-HPLC method


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232176
PNG
(CHEMBL4091749)
Show SMILES Oc1ccc(F)c(C(=O)c2ccc(s2)-c2cc(Cl)c(O)c(Cl)c2)c1F
Show InChI InChI=1S/C17H8Cl2F2O3S/c18-8-5-7(6-9(19)16(8)23)12-3-4-13(25-12)17(24)14-10(20)1-2-11(22)15(14)21/h1-6,22-23H
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n/an/a 2.40n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Estradiol 17-beta-dehydrogenase 1


(Homo sapiens (Human))
BDBM50232165
PNG
(CHEMBL4067584)
Show SMILES NS(=O)(=O)c1cccc(c1)-c1ccc(s1)C(=O)c1c(F)ccc(O)c1F
Show InChI InChI=1S/C17H11F2NO4S2/c18-11-4-5-12(21)16(19)15(11)17(22)14-7-6-13(25-14)9-2-1-3-10(8-9)26(20,23)24/h1-8,21H,(H2,20,23,24)
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n/an/a 55n/an/an/an/an/an/a



Saarland University

Curated by ChEMBL


Assay Description
Inhibition of human placental cytosolic 17beta-HSD1 assessed as reduction in activation of [2,4,6,7-3H]-E1 substrate to E2 after 10 mins in presence ...


Eur J Med Chem 127: 944-957 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.004
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM50232205
PNG
(CHEMBL4080865)
Show SMILES CCCc1nc2ccc(cc2n1Cc1ccc(cc1)-c1ccccc1C(O)=O)-c1ccc(Cl)cc1
Show InChI InChI=1S/C30H25ClN2O2/c1-2-5-29-32-27-17-14-23(21-12-15-24(31)16-13-21)18-28(27)33(29)19-20-8-10-22(11-9-20)25-6-3-4-7-26(25)30(34)35/h3-4,6-18H,2,5,19H2,1H3,(H,34,35)
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n/an/an/an/a 1.15E+3n/an/an/an/a



University of Innsbruck

Curated by ChEMBL


Assay Description
Transactivation of Gal4 fused human PPARgamma LBD expressed in African green monkey COS7 cells after 42 hrs by dual luciferase reporter gene assay


Eur J Med Chem 126: 590-603 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.051
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM50232210
PNG
(CHEMBL4078107)
Show SMILES CCCc1nc2cc(ccc2n1Cc1ccc(cc1)-c1ccccc1C(O)=O)-c1cccc(OC)c1
Show InChI InChI=1S/C31H28N2O3/c1-3-7-30-32-28-19-24(23-8-6-9-25(18-23)36-2)16-17-29(28)33(30)20-21-12-14-22(15-13-21)26-10-4-5-11-27(26)31(34)35/h4-6,8-19H,3,7,20H2,1-2H3,(H,34,35)
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n/an/an/an/a 290n/an/an/an/a



University of Innsbruck

Curated by ChEMBL


Assay Description
Transactivation of Gal4 fused human PPARgamma LBD expressed in African green monkey COS7 cells after 42 hrs by dual luciferase reporter gene assay


Eur J Med Chem 126: 590-603 (2017)


Article DOI: 10.1016/j.ejmech.2016.11.051
More data for this
Ligand-Target Pair
Estrogen-related receptor alpha


(Homo sapiens (Human))
BDBM50232198
PNG
(CHEMBL4095236)
Show SMILES C[C@@H]1CN(CCN1c1ccc(cn1)C(C)=O)C(=O)c1cc2c(C)nn(Cc3cccc(OCCCCNC(=O)CCC4=[N+]5C(C=C4)=Cc4c(C)cc(C)n4[B-]5(F)F)c3)c2s1
Show InChI InChI=1S/C44H49BF2N8O4S/c1-28-21-29(2)54-39(28)23-36-13-12-35(55(36)45(54,46)47)14-16-42(57)48-17-6-7-20-59-37-10-8-9-33(22-37)27-53-44-38(31(4)50-53)24-40(60-44)43(58)51-18-19-52(30(3)26-51)41-15-11-34(25-49-41)32(5)56/h8-13,15,21-25,30H,6-7,14,16-20,26-27H2,1-5H3,(H,48,57)/t30-/m1/s1
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n/an/a 170n/an/an/an/an/an/a



Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL


Assay Description
Inverse agonist activity at GAL4-fused human ERRalpha expressed in HEK293 cells assessed as inhibition of transcriptional activity after 20 hrs by lu...


Bioorg Med Chem Lett 27: 1145-1148 (2017)


Article DOI: 10.1016/j.bmcl.2017.01.076
More data for this
Ligand-Target Pair