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There are 2 purchasable compounds for target: Prokineticin receptor 2 (PRK2)

Compile data set for download or QSAR
Wt: 144.2
BDBM121028
Purchase
Wt: 144.2
BDBM121337
Purchase

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 121028,121337   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Prokineticin receptor 2 (PRK2)


(Cricetulus griseus (Chinese hamster))
BDBM121028
PNG
(US8722896, (+)-(2S)-2-Amino-N- isobutylpropanamide)
Show SMILES CC(C)CNC(=O)C(C)N
Show InChI InChI=1/C7H16N2O/c1-5(2)4-9-7(10)6(3)8/h5-6H,4,8H2,1-3H3,(H,9,10)
UniProtKB/TrEMBL

GoogleScholar
Purchase

PC cid
PC sid
UniChem

Similars

US Patent
9.84E+3 -7.10n/an/an/an/an/an/a37



The Regents of the University of California

US Patent


Assay Description
An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...


US Patent US8722896 (2014)


BindingDB Entry DOI: 10.7270/Q29G5KGF
More data for this
Ligand-Target Pair
Prokineticin receptor 2 (PRK2)


(Cricetulus griseus (Chinese hamster))
BDBM121337
PNG
(US8722896, (-)-(2R)-2-Amino-N- isobutylpropanamide)
Show SMILES CC(C)CNC(=O)[C@H](C)N
Show InChI InChI=1/C7H16N2O/c1-5(2)4-9-7(10)6(3)8/h5-6H,4,8H2,1-3H3,(H,9,10)/t6-/s2
UniProtKB/TrEMBL

GoogleScholar
Purchase

KEGG
PC cid
PC sid
UniChem

Similars

US Patent
>1.00E+4>-7.09n/an/an/an/an/an/a37



The Regents of the University of California

US Patent


Assay Description
An aequorin-based luminescent assay for calcium mobilization was used to measure mobilization of intracellular Ca2+ (Bullock et al., Mol Pharmacol 65...


US Patent US8722896 (2014)


BindingDB Entry DOI: 10.7270/Q29G5KGF
More data for this
Ligand-Target Pair