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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50128081(CHEMBL2369390 | Tyr-Gly-Pro-Phe-Leu-Arg-Arg-Ile-NH...)
Affinity DataKi:  10.7nMAssay Description:In vitro binding affinity to human Opioid receptor mu 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50128081(CHEMBL2369390 | Tyr-Gly-Pro-Phe-Leu-Arg-Arg-Ile-NH...)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity towards human Opioid receptor kappa 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50128081(CHEMBL2369390 | Tyr-Gly-Pro-Phe-Leu-Arg-Arg-Ile-NH...)
Affinity DataKi:  1.32E+4nMAssay Description:In vitro binding affinity to human Opioid receptor delta 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed