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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Affinity Data
Ki: 6.80nM
Assay Description:
Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
Allergan
Curated by
ChEMBL
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Affinity Data
Ki: 9.60nM
Assay Description:
Compound was tested in vitro for binding affinity against Alpha-2A adrenergic receptor from cloned human C-10 receptor transfected into Chinese hamst...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
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Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Copy InChI
Affinity Data
Ki: 9.60nM
Assay Description:
Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Copy BDB DOI
Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
Allergan
Curated by
ChEMBL
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Copy InChI
Affinity Data
Ki: 120nM
Assay Description:
Compound was tested in vitro for binding affinity against Alpha-2C adrenergic receptor from cloned human C-2 receptor transfected into Chinese hamste...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Alpha-2B adrenergic receptor
(NEONATAL RAT)
Allergan
Curated by
ChEMBL
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Affinity Data
Ki: 140nM
Assay Description:
Compound was tested in vitro for binding affinity against Alpha-2B adrenergic receptor from cloned rat RNG receptor transfected into Chinese hamster ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Affinity Data
Ki: 8.70E+3nM
Assay Description:
Binding affinity towards Alpha-1 adrenergic receptor in human brain
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Copy BDB DOI
Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50052881
(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
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Affinity Data
Ki: 8.90E+3nM
Assay Description:
Binding affinity for Alpha-1 adrenergic receptor of human cerebral cortex membrane
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Copy BDB DOI