Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50346316((S)-2-(phenylsulfonamido)-3-(4-((S)-3-(1,4,5,6-tet...)
Affinity DataIC50:  0.480nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50346316((S)-2-(phenylsulfonamido)-3-(4-((S)-3-(1,4,5,6-tet...)
Affinity DataIC50:  0.560nMAssay Description:Antagonist activity at alpha2bbeta3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50346316((S)-2-(phenylsulfonamido)-3-(4-((S)-3-(1,4,5,6-tet...)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed