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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProtein kinase YpkA(Yersinia pestis)
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50:  5.87E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50:  5.30E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Rockefeller University

LigandPNGBDBM22045(5-({4-[(4-chlorophenyl)sulfanyl]-3-nitrophenyl}met...)
Affinity DataIC50: >2.00E+5nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed for autophosphorylation and phosphorylation of MBP with radio-labeled gamma-32P. IC50 values were calculated from binding...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed