Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 4 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonistic activity against mouse Melanocortin 1 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed