Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001323(16,24-dibenzyl-25-methyl-13-[1-methyl-(1S)-propyl]...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of [3H]arginine vasopressin binding to AVP-V2 site in rat kidney medulla.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001323(16,24-dibenzyl-25-methyl-13-[1-methyl-(1S)-propyl]...)
Affinity DataIC50:  3.50E+3nMAssay Description:Concentration required to displace 50% of [3H]arginine vasopressin from rat liver arginine vasopressin 1A (AVP-V1a) site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50001323(16,24-dibenzyl-25-methyl-13-[1-methyl-(1S)-propyl]...)
Affinity DataIC50:  3.50E+3nMAssay Description:Concentration required to displace 50% of [3H]oxytocin from rat uterine receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed