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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNicotinic acetylcholine receptor alpha9/alpha10(RAT)
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50032829(CHEMBL1836968)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of rat alpha9alpha10 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor; alpha9/alpha10(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50032829(CHEMBL1836968)
Affinity DataIC50:  510nMAssay Description:Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response by two-e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50032829(CHEMBL1836968)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human alpha7 nAChR expressed in Xenopus oocytes assessed as inhibition of Ach-evoked current after 5 mins by voltage-clamp techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Ocean University Of China

Curated by ChEMBL
LigandPNGBDBM50032829(CHEMBL1836968)
Affinity DataIC50:  4.66E+3nMAssay Description:Inhibition of rat alpha7 nAChRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed