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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50228680(CHEMBL345810)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in rat cerebral cortical membrane using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228680(CHEMBL345810)
Affinity DataKi:  251nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in rat cerebral cortical membrane using [3H]yohimbine as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed