Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
Neuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))Glaxo Wellcome Research And Development
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
IC50: 180nMAssay Description:Inhibition of influenza sialidase was determined by measuring the ability to inhibit the hydrolysis of MUN by A/Aichi virus grown in hen eggsMore data for this Ligand-Target Pair
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
IC50: 2.30E+4nMAssay Description:Inhibition of influenza sialidase was determined by measuring the ability to inhibit the hydrolysis of MUN by B Victoria virus grown in hen eggsMore data for this Ligand-Target Pair
Neuraminidase(Influenza B virus)Glaxo Wellcome Research And Development
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
IC50: 2.30E+4nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
BDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)