Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50122993(CHEMBL2370452 | [(1R,18S,19R,20S)-14-(3-Guanidino-...)
Affinity DataIC50:  3.22E+4nMAssay Description:Displacement of [125I]-echistatin from alphaIIb-beta3 integrin of human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50122993(CHEMBL2370452 | [(1R,18S,19R,20S)-14-(3-Guanidino-...)
Affinity DataIC50:  9.81E+4nMAssay Description:Displacement of [125I]-echistatin from alphaV-beta3 integrin of human skin fibroblastsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed