Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
Ki: 83.1nMAssay Description:Binding affinity measured on Sigma receptor type 1 from guinea pig brain membranes using [3H]pentazocine as radioligand.More data for this Ligand-Target Pair
BDBM50001033((-)-Pentazocine | 3-But-2-enyl-6,11-dimethyl-1,2,3...)
IC50: 8.90nMAssay Description:Compound was evaluated for the binding affinity towards Sigma receptor type 1 using radioligand ([3H]-(+)- Pentazocine) binding assay.More data for this Ligand-Target Pair
IC50: 29nMAssay Description:Binding affinity towards Sigma receptor type 2 in whole rat brain homogenates except cerebellum using radioligand ([3H]DTG) binding assay.More data for this Ligand-Target Pair