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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Muscarinic acetylcholine receptor M1
(RAT)
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM50454824
(CHEMBL3084909)
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Affinity Data
Ki: 0.850nM
Assay Description:
Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM50454824
(CHEMBL3084909)
Copy SMILES
Copy InChI
Affinity Data
Ki: 47nM
Assay Description:
Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate Putamen
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM50454824
(CHEMBL3084909)
Copy SMILES
Copy InChI
Affinity Data
Ki: 48nM
Assay Description:
Binding affinity to dopamine transporter (DAT) using [3H]WIN-35428 as a radioligand
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Sodium-dependent dopamine transporter
(Rattus norvegicus (rat))
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM50454824
(CHEMBL3084909)
Copy SMILES
Copy InChI
Affinity Data
IC50: 407nM
Assay Description:
[3H]-Dopamine uptake inhibition in rat caudate putamen
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI