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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSteroidogenic factor 1(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22384((3aS,6aR)-5-methyl-N,4-diphenyl-1,2,3,3a,6,6a-hexa...)
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton

LigandPNGBDBM22384((3aS,6aR)-5-methyl-N,4-diphenyl-1,2,3,3a,6,6a-hexa...)
Affinity DataEC50:  2.10E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed