Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

LigandPNGBDBM50229152(CHEMBL349004)
Affinity DataKi:  0.708nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50229152(CHEMBL349004)
Affinity DataKi:  1.29E+4nMAssay Description:Binding affinity to alpha-1 adrenergic receptor determined by measurement of [3H]prazosin displacement from rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed