Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
Kd: 1.38E+3nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
Kd: 1.66E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
BDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)