Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Monoglyceride lipase
(Mus musculus (mouse))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 200nM
Assay Description:
Inhibition of MAGL in mouse brain membrane
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Monoglyceride lipase
(Mus musculus (mouse))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 282nM
Assay Description:
Inhibition of mouse MAGL
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Monoglyceride lipase
(Homo sapiens (Human))
University Of Eastern Finland
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 347nM
Assay Description:
Inhibition of human recombinant MAGL expressed in HEK293 cells using 2-AG as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Monoacylglycerol lipase ABHD6
(Mus musculus (mouse))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 900nM
Assay Description:
Inhibition of ABHD6 in mouse brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Monoglyceride lipase
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.80E+3nM
Assay Description:
Inhibition of rat MAGL
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Fatty-acid amide hydrolase 1
(Mus musculus (mouse))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50307064
(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.41E+3nM
Assay Description:
Inhibition of FAAH in mouse brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI