Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetMonoglyceride lipase(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  200nMAssay Description:Inhibition of MAGL in mouse brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  282nMAssay Description:Inhibition of mouse MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  347nMAssay Description:Inhibition of human recombinant MAGL expressed in HEK293 cells using 2-AG as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoacylglycerol lipase ABHD6(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  900nMAssay Description:Inhibition of ABHD6 in mouse brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50307064(4-nitrophenyl 4-(bis(4-fluorophenyl)methyl)piperaz...)
Affinity DataIC50:  5.41E+3nMAssay Description:Inhibition of FAAH in mouse brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed