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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50223673(5-nitro-N-(2-(pyrrolidin-1-yl)phenyl)furan-2-carbo...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of ATP-induced autophosphorylation of cFMS tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSentrin-specific protease 8(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM50223673(5-nitro-N-(2-(pyrrolidin-1-yl)phenyl)furan-2-carbo...)
Affinity DataIC50:  6.69E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSentrin-specific protease 8(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM50223673(5-nitro-N-(2-(pyrrolidin-1-yl)phenyl)furan-2-carbo...)
Affinity DataIC50:  6.69E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay